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1 . Academic Journal
Dose-dependent effects of GAT107, a novel allosteric agonist-positive allosteric modulator (ago-PAM) for the α7 nicotinic cholinergic receptor: a BOLD phMRI and connectivity study on awake rats
저자
by
Brittany M. Brems
;
Erin E. Sullivan
;
Jenna G. Connolly
;
Jingchun Zhang
;
Arnold Chang
, et al.
소스
Frontiers in Neuroscience, Vol 17 (2023)
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7 . Academic Journal
The type 1 cannabinoid receptor positive allosteric modulators GAT591 and GAT593 reduce spike-and-wave discharges in Genetic Absence Epilepsy Rats from Strasbourg
저자
by
Dan L. McElroy
;
Andrew J. Roebuck
;
Quentin Greba
;
Sumanta Garai
;
Asher L. Brandt
, et al.
소스
IBRO Neuroscience Reports, Vol 12, Iss , Pp 121-130 (2022)
Full Text (ScienceDirect)
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7 . Academic Journal
Pharmacological evaluation of enantiomerically separated positive allosteric modulators of cannabinoid 1 receptor, GAT591 and GAT593
저자
by
Asher L. Brandt
;
Sumanta Garai
;
Ayat Zagzoog
;
Dow P. Hurst
;
Lesley A. Stevenson
, et al.
소스
Frontiers in Pharmacology, Vol 13 (2022)
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7 . Academic Journal
Suppression of neuroinflammation by an allosteric agonist and positive allosteric modulator of the α7 nicotinic acetylcholine receptor GAT107
저자
by
Tehila Mizrachi
;
Oshrit Marsha
;
Karen Brusin
;
Yael Ben-David
;
Ganesh A. Thakur
, et al.
소스
Journal of Neuroinflammation, Vol 18, Iss 1, Pp 1-14 (2021)
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7 . Academic Journal
Use of a Molecular Switch Probe to Activate or Inhibit GIRK1 Heteromers In Silico Reveals a Novel Gating Mechanism
저자
by
Dimitrios Gazgalis
;
Lucas Cantwell
;
Yu Xu
;
Ganesh A. Thakur
;
Meng Cui
, et al.
소스
International Journal of Molecular Sciences, Vol 23, Iss 18, p 10820 (2022)
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7 . Academic Journal
Peripheral versus central mechanisms of the cannabinoid type 2 receptor agonist AM1710 in a mouse model of neuropathic pain
저자
by
Jenny L. Wilkerson
;
Lauren B. Alberti
;
Audra A. Kerwin
;
Catherine A. Ledent
;
Ganesh A. Thakur
, et al.
소스
Brain and Behavior, Vol 10, Iss 12, Pp n/a-n/a (2020)
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7 . Academic Journal
Positive Allosteric Modulation of CB1 Cannabinoid Receptor Signaling Enhances Morphine Antinociception and Attenuates Morphine Tolerance Without Enhancing Morphine- Induced Dependence or Reward
저자
by
Richard A. Slivicki
;
Vishakh Iyer
;
Sonali S. Mali
;
Sumanta Garai
;
Ganesh A. Thakur
, et al.
소스
Frontiers in Molecular Neuroscience, Vol 13 (2020)
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7 . Academic Journal
Indomethacin Enhances Type 1 Cannabinoid Receptor Signaling
저자
by
Robert B. Laprairie
;
Kawthar A. Mohamed
;
Ayat Zagzoog
;
Melanie E. M. Kelly
;
Lesley A. Stevenson
, et al.
소스
Frontiers in Molecular Neuroscience, Vol 12 (2019)
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7 . Academic Journal
The Positive Allosteric Modulation of alpha7-Nicotinic Cholinergic Receptors by GAT107 Increases Bacterial Lung Clearance in Hyperoxic Mice by Decreasing Oxidative Stress in Macrophages
저자
by
Alex G. Gauthier
;
Jiaqi Wu
;
Mosi Lin
;
Ravikumar Sitapara
;
Abhijit Kulkarni
, et al.
소스
Antioxidants, Vol 10, Iss 1, p 135 (2021)
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7 . Academic Journal
Allosteric Cannabinoid Receptor 1 (CB1) Ligands Reduce Ocular Pain and Inflammation
저자
by
Dinesh Thapa
;
Elizabeth A. Cairns
;
Anna-Maria Szczesniak
;
Pushkar M. Kulkarni
;
Alex J. Straiker
, et al.
소스
Molecules, Vol 25, Iss 2, p 417 (2020)
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