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1 . Academic Journal
Synthesis and Structure–Activity Relationship of C-Phenyl D-Glucitol (TP0454614) Derivatives as Selective Sodium-Dependent Glucose Cotransporter 1 (SGLT1) Inhibitors
저자
by
Fumiyasu Shiozawa
;
Hiroko Koretsune
;
Hiroyuki Kakinuma
;
Kayo Kimura
;
Kenichi Kawabe
, et al.
소스
Chemical and Pharmaceutical Bulletin. 2020, 68(7):635
Open Access (JSTAGE)
Web of Science
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7 .
Discovery of potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor SGL5213 for type 2 diabetes treatment
저자
by
Mami Sugisaki-Kitano
;
Takahiro Oi
;
Lisa Okumura-Kitajima
;
Fumiyasu Shiozawa
;
Yohei Kobashi
, et al.
소스
Bioorganic & Medicinal Chemistry
. 27:394-409
Web of Science
Scopus
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7 .
Synthesis and Structure-Activity Relationship of C-Phenyl D-Glucitol (TP0454614) Derivatives as Selective Sodium-Dependent Glucose Cotransporter 1 (SGLT1) Inhibitors
저자
by
Hiroyuki Kakinuma
;
Yuki Shimizu
;
Kayo Kimura
;
Yohei Kobashi
;
Lisa Okumura-Kitajima
, et al.
소스
Chemicalpharmaceutical bulletin
. 68(7)
Open Access (OpenAIRE)
Scopus
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7 .
Design, synthesis and biological evaluation of novel 7-azaspiro[3.5]nonane derivatives as GPR119 agonists
저자
by
Norikazu Ohtake
;
Keiko Fusegi
;
Fumiyasu Shiozawa
;
Masako Miyoshi
;
Madoka Kawamura
, et al.
소스
Bioorganic & Medicinal Chemistry
. 26:1832-1847
Web of Science
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7 .
Design and synthesis of 1H-pyrazolo[3,4-c]pyridine derivatives as a novel structural class of potent GPR119 agonists
저자
by
Madoka Kawamura
;
Masako Miyoshi
;
Fumiyasu Shiozawa
;
Yohei Kobashi
;
Kayo Kimura
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 26:3441-3446
Web of Science
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7 .
Lymphopenia induced by a novel selective S1P1 antagonist structurally unrelated to S1P
저자
by
Ryo Goitsuka
;
Takehiro Hirayama
;
Tetsuo Takayama
;
Takanobu Sakurai
;
Yasuyuki Igarashi
, et al.
소스
Biochimica et Biophysica Acta (BBA) - Molecular and Cell Biology of Lipids
. 1821:600-606
Web of Science
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7 .
Pyrrole derivatives as potent inhibitors of lymphocyte-specific kinase: Structure, synthesis, and SAR
저자
by
Tetsuo Takayama
;
Tetsuya Yabuuchi
;
Hironori Katakai
;
Mayumi Endo
;
Akiko Takaoka
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 20:108-111
Web of Science
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7 .
Ring-fused pyrazole derivatives as potent inhibitors of lymphocyte-specific kinase (Lck): Structure, synthesis, and SAR
저자
by
Hiroki Umemiya
;
Yusuke Oka
;
Fumiyasu Shiozawa
;
Akiko Takaoka
;
Hideaki Amada
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 20:112-116
Web of Science
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7 .
Synthesis of Isochromene Esters Utilizing 1,6-Addition of Nucleophiles to Benzopyranylidenetungsten(0) Complexes
저자
by
Fumiyasu Shiozawa
;
Hiroyuki Kusama
;
Atsushi Okita
;
Takahiro Sawada
;
Nobuharu Iwasawa
.
소스
Org. Lett.
. 8:1077-7079
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7 .
Design, synthesis, and evaluation of novel 4-thiazolylimidazoles as inhibitors of transforming growth factor-β type I receptor kinase
저자
by
Masakazu Sato
;
Fumiyasu Shiozawa
;
Mari Aoki
;
Naoya Ono
;
Natsuko Fujimoto
, et al.
소스
Bioorganicmedicinal chemistry letters
. 22(5)
Full Text (ScienceDirect)
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