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1 . Academic Journal
Creating a more strategic small molecule biophysical hit characterization workflow
저자
by
Fotsch, Christopher
;
Basu, Debaleena
;
Case, Ryan
;
Chen, Qing
;
Koneru, Pratibha C.
, et al.
소스
In
SLAS Discovery
June 2024 29(4)
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7 . Academic Journal
On-resin macrocyclization of peptides via intramolecular S nAr reactions
저자
by
Fotsch, Christopher
;
Kumaravel, G.
;
Sharma, Sushil K.
;
Wu, Arthur D.
;
Gounarides, John S.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1999 9(15):2125-2130
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7 . Academic Journal
The optimization of aminooxadiazoles as orally active inhibitors of Cdc7
저자
by
Harrington, Paul E.
;
Bourbeau, Matthew P.
;
Fotsch, Christopher
;
Frohn, Michael
;
Pickrell, Alexander J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2013 23(23):6396-6400
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7 . Academic Journal
Systematic Study of the Glutathione Reactivity of N‑Phenylacrylamides: 2. Effects of Acrylamide Substitution.
저자
by
Birkholz, Adam
;
Kopecky, David J.
;
Volak, Laurie P.
;
Bartberger, Michael D.
;
Chen, Yuping
, et al.
소스
Journal of Medicinal Chemistry; 10/22/2020, Vol. 63 Issue 20, p11602-11614, 13p
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7 . Academic Journal
Quinolinone-based agonists of S1P1: Use of a N-scan SAR strategy to optimize in vitro and in vivo activity
저자
by
Pennington, Lewis D.
;
Croghan, Michael D.
;
Sham, Kelvin K.C.
;
Pickrell, Alexander J.
;
Harrington, Paul E.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 January 2012 22(1):527-531
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7 . Academic Journal
Design and synthesis of novel amide AKT1 inhibitors with selectivity over CDK2
저자
by
Ashton, Kate S.
;
St. Jean, David J., Jr.
;
Poon, Steve F.
;
Lee, Matthew R.
;
Allen, John G.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 September 2011 21(18):5191-5196
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7 . Academic Journal
3-Oxo-2-piperazinyl acetamides as potent bradykinin B1 receptor antagonists for the treatment of pain and inflammation
저자
by
Chen, Jian Jeffrey
;
Nguyen, Thomas
;
D’Amico, Derin C.
;
Qian, Wenyuan
;
Human, Jason
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(11):3384-3389
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7 . Academic Journal
Aryl sulfonamides containing tetralin allylic amines as potent and selective bradykinin B1 receptor antagonists
저자
by
Liu, Qingyian
;
Qian, Wenyuan
;
Li, Aiwen
;
Biswas, Kaustav
;
Chen, Jian Jeffrey
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2010 20(15):4593-4597
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7 . Academic Journal
The discovery of an orally efficacious positive allosteric modulator of the calcium sensing receptor containing a dibenzylamine core
저자
by
Harrington, Paul E.
;
St. Jean, David J., Jr.
;
Clarine, Jeffrey
;
Coulter, Thomas S.
;
Croghan, Michael
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(18):5544-5547
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7 . Academic Journal
Azole-based inhibitors of AKT/PKB for the treatment of cancer
저자
by
Zeng, Qingping
;
Allen, John G.
;
Bourbeau, Matthew P.
;
Wang, Xianghong
;
Yao, Guomin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(5):1559-1564
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