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1 . Academic Journal
Identification of MK-5710 ((8 aS)-8 a-methyl-1,3-dioxo-2-[(1 S,2 R)-2-phenylcyclo- propyl]- N-(1-phenyl-1 H-pyrazol-5-yl)hexahydro-imidazo[1,5- a]pyrazine-7(1 H)-carboxamide), a potent smoothened antagonist for use in Hedgehog pathway dependent malignancies, Part 2
저자
by
Kinzel, Olaf
;
Alfieri, Anna
;
Altamura, Sergio
;
Brunetti, Mirko
;
Bufali, Simone
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(15):4429-4435
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7 . Academic Journal
Identification of MK-5710 ((8 aS)-8 a-methyl-1,3-dioxo-2-[(1 S,2 R)-2-phenylcyclopropyl]- N-(1-phenyl-1 H-pyrazol-5-yl)hexahydroimid azo[1,5-a]pyrazine-7(1 H)-carboxamide), a potent smoothened antagonist for use in Hedgehog pathway dependent malignancies, Part 1
저자
by
Malancona, Savina
;
Altamura, Sergio
;
Filocamo, Gessica
;
Kinzel, Olaf
;
Hernando, Jose Ignacio Martin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(15):4422-4428
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7 .
Efficacy of selective histone deacetylase 6 inhibition in mouse models of Pseudomonas aeruginosa infection. A new glimpse for reducing inflammation and infection in cystic fibrosis
저자
by
Margherita Brindisi
;
Simona Barone
;
Alice Rossi
;
Emilia Cassese
;
Nunzio Del Gaudio
, et al.
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7 . Academic Journal
Efficacy of selective histone deacetylase 6 inhibition in mouse models of Pseudomonas aeruginosa infection: A new glimpse for reducing inflammation and infection in cystic fibrosis.
저자
by
Brindisi, Margherita
;
Barone, Simona
;
Rossi, Alice
;
Cassese, Emilia
;
Del Gaudio, Nunzio
, et al.
소스
European Journal of Pharmacology
. Dec2022, Vol. 936, pN.PAG-N.PAG. 1p.
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7 . Academic Journal
Dissecting the Biological Functions of Drosophila Histone Deacetylases by RNA Interference and Transcriptional ProfiIing.
저자
by
Fogiietti, Cristiana
;
Filocamo, Gessica
;
Cundari, Enrico
;
De Rinaldis, Emanuele
;
Lahm, Armin
, et al.
소스
Journal of Biological Chemistry
. 6/30/2006, Vol. 281 Issue 26, p17968-17976. 9p. 2 Diagrams, 1 Chart, 6 Graphs.
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7 . Academic Journal
Crystal structure of a eukaryotic zinc-dependent histone deacetylase, human HDAC8, complexed with a hydroxamic acid inhibitor.
저자
by
Vannini, Alessandro
;
Volpari, Cinzia
;
Filocamo, Gessica
;
Casavola, Elena Caroli
;
Brunetti, Mirko
, et al.
소스
Proceedings of the National Academy of Sciences of the United States of America
. 10/19/2004, Vol. 101 Issue 42, p15064-15069. 6p.
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7 . Academic Journal
The human scavenger receptor class B type I is a novel candidate receptor for the hepatitis C virus.
저자
by
Scarselli, Elisa
;
Ansuini, Helenia
;
Cerino, Raffaele
;
Roccasecca, Rosa Maria
;
Acali, Stefano
, et al.
소스
EMBO Journal
. 10/1/2002, Vol. 21 Issue 19, p5017-5025. 9p.
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7 . Periodical
Smoothened antagonists: a promising new class of antitumor agents
저자
by
Gallinari, Paola
;
Filocamo, Gessica
;
Jones, Philip
;
Pazzaglia, Simonetta
;
Steinkühler, Christian
.
소스
Expert Opinion on Drug Discovery; January 2009, Vol. 4 Issue: 5 p525-544, 20p
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7 . Periodical
In Vivo Selection of Protease Cleavage Sites by Using Chimeric Sindbis Virus Libraries
저자
by
Pacini, Laura
;
Vitelli, Alessandra
;
Filocamo, Gessica
;
Bartholomew, Linda
;
Brunetti, Mirko
, et al.
소스
The Journal of Virology; November 2000, Vol. 74 Issue: 22 p10563-10570, 8p
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7 . Periodical
Selection of Functional Variants of the NS3-NS4A Protease of Hepatitis C Virus by Using Chimeric Sindbis Viruses
저자
by
Filocamo, Gessica
;
Pacini, Laura
;
Nardi, Chiara
;
Bartholomew, Linda
;
Scaturro, Maria
, et al.
소스
The Journal of Virology; January 1999, Vol. 73 Issue: 1 p561-575, 15p
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