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1 .
Discovery of Selective Pituitary Adenylate Cyclase 1 Receptor (PAC1R) Antagonist Peptides Potent in a Maxadilan/PACAP38-Induced Increase in Blood Flow Pharmacodynamic Model
저자
by
Fang-Tsao Hong
;
Hongyan Li
;
Derek E. Piper
;
Leszek Poppe
;
Philip Wong
, et al.
소스
Journal of Medicinal Chemistry
. 64:3427-3438
Web of Science
Scopus
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7 .
Abstract LB318: SB-4826, a first-in-class oral, covalent inhibitor of SUMO E1 that induces IFN signaling and inhibits tumor growth as monotherapy and in combination with immune checkpoint blockade
저자
by
Jude R. Canon
;
Ashley Callinan
;
Sarah Bradley
;
Laurie Wang
;
Mackenzie Kui
, et al.
소스
Cancer Research
. 83:LB318-LB318
Full Text (AACR)
Web of Science
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7 . Academic Journal
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase-Glucokinase Regulatory Protein (GK-GKRP) Binding: Strategic Use of a N → S (n
N
→ s*
S-X
) Interaction for Conformational Constraint
저자
by
Pennington, Lewis D.
;
Bartberger, Michael D.
;
Croghan, Michael D.
;
Andrews, Kristin L.
;
Ashton, Kate S.
, et al.
소스
Journal of Medicinal Chemistry
. Dec2015, Vol. 58 Issue 24, p9663-9679. 17p.
Full Text (ACS)
Web of Science
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7 . Academic Journal
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase-Glucokinase Regulatory Protein (GK-GKRP) Binding: Strategic Use of a N → S (n
N
→ s*
S-X
) Interaction for Conformational...
저자
by
Pennington, Lewis D.
;
Bartberger, Michael D.
;
Croghan, Michael D.
;
Andrews, Kristin L.
;
Ashton, Kate S.
, et al.
소스
Journal of Medicinal Chemistry; Dec2015, Vol. 58 Issue 24, p9663-9679, 17p
Full Text (ACS)
Web of Science
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7 . Academic Journal
Small Molecule Disruptors of the Glucokinase–GlucokinaseRegulatory Protein Interaction: 5. A Novel Aryl Sulfone Series, OptimizationThrough Conformational Analysis.
저자
by
Nuria A. Tamayo
;
Mark H. Norman
;
Michael D. Bartberger
;
Fang-Tsao Hong
;
Yunxin Bo
, et al.
소스
Journal of Medicinal Chemistry
. Jun2015, Vol. 58 Issue 11, p4462-4482. 21p.
Full Text (ACS)
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7 . Academic Journal
Total Synthesis of Dumsin. 1. Retrosynthetic Strategy and the Elaboration of Key Intermediates from (-)-Bornyl Acetate.
저자
by
Paquette, Leo A.
;
Fang-Tsao Hong
.
소스
Journal of Organic Chemistry
. 9/5/2003, Vol. 68 Issue 18, p6905-6918. 14p. 22 Diagrams.
Full Text (ACS)
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4 . Academic Journal
Stereocontrolled Synthesis of Triazacyclopental[cd]pentalenes by Intramolecular 1,3-Dipolar Cycloaddition Reactions of Azomethine Imines.
저자
by
Bélanger, Guillaume
;
Fang-Tsao Hong
;
Overman, Larry E.
;
Rogers, Bruce N.
;
Tellew, John E.
, et al.
소스
Journal of Organic Chemistry
. 11/1/2002, Vol. 67 Issue 22, p7880. 4p. 5 Diagrams.
Full Text (ACS)
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7 . Academic Journal
Heteroatomic effects on the reducibility of C-2 carbinol centers in 6-ethoxy-3,6-dihydropyrans...
저자
by
Fang-Tsao Hong
;
Paquette, Leo A.
.
소스
Journal of Organic Chemistry
. 05/14/99, Vol. 64 Issue 10, p3783. 4p. 4 Diagrams.
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4 .
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase–Glucokinase Regulatory Protein (GK–GKRP) Binding: Strategic Use of a N → S (nN → σ*S–X) Interaction for Conformational Constraint
저자
by
Michael D. Bartberger
;
Michael Croghan
;
Carolyn Moyer
;
David Lloyd
;
Rod Cupples
, et al.
소스
Journal of Medicinal Chemistry
. 58:9663-9679
Open Access (OpenAIRE)
Web of Science
Scopus
JCR 저널정보
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RefWorks
7 .
Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 5. A Novel Aryl Sulfone Series, Optimization Through Conformational Analysis
저자
by
Kevin Yang
;
Rod Cupples
;
Gwyneth Van
;
Nobuko Nishimura
;
Longbin Liu
, et al.
소스
Journal of Medicinal Chemistry
. 58:4462-4482
Web of Science
Scopus
JCR 저널정보
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