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1 . Academic Journal
Discovery, synthesis, and structure-activity relations of 3,4-dihydro-1H-spiro(naphthalene-2,2′-piperidin)-1-ones as potassium-competitive acid blockers
저자
by
Imaeda, Toshihiro
;
Ono, Koji
;
Nakai, Kazuo
;
Hori, Yasunobu
;
Matsukawa, Jun
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 July 2017 25(14):3719-3735
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7 . Academic Journal
Identification of a novel fluoropyrrole derivative as a potassium-competitive acid blocker with long duration of action
저자
by
Nishida, Haruyuki
;
Arikawa, Yasuyoshi
;
Hirase, Keizo
;
Imaeda, Toshihiro
;
Inatomi, Nobuhiro
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 July 2017 25(13):3298-3314
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7 . Academic Journal
Exploration of pyrrole derivatives to find an effective potassium-competitive acid blocker with moderately long-lasting suppression of gastric acid secretion
저자
by
Nishida, Haruyuki
;
Fujimori, Ikuo
;
Arikawa, Yasuyoshi
;
Hirase, Keizo
;
Ono, Koji
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 July 2017 25(13):3447-3460
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7 . Academic Journal
Design, synthesis, and biological evaluation of a novel series of peripheral-selective noradrenaline reuptake inhibitors – Part 3
저자
by
Yukawa, Tomoya
;
Nakada, Yoshihisa
;
Sakauchi, Nobuki
;
Kamei, Taku
;
Yamada, Masami
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 August 2016 24(16):3716-3726
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7 . Academic Journal
Design, synthesis, and biological evaluation of a novel series of peripheral-selective noradrenaline reuptake inhibitors—Part 2
저자
by
Yukawa, Tomoya
;
Fujimori, Ikuo
;
Kamei, Taku
;
Nakada, Yoshihisa
;
Sakauchi, Nobuki
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 July 2016 24(14):3207-3217
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7 . Academic Journal
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibition
저자
by
Igawa, Hideyuki
;
Takahashi, Masashi
;
Shirasaki, Mikio
;
Kakegawa, Keiko
;
Kina, Asato
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 June 2016 24(11):2486-2503
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7 . Academic Journal
Evaluation of Acid Tolerance of Drugs Using Rats and Dogs Controlled for Gastric Acid Secretion
저자
by
Kosugi, Yohei
;
Yamamoto, Syunsuke
;
Sano, Noriyasu
;
Furuta, Atsutoshi
;
Igari, Tomoko
, et al.
소스
In
Journal of Pharmaceutical Sciences
September 2015 104(9):2887-2893
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7 . Academic Journal
Establishment and Validation of a Rabbit Model for In Vivo Pharmacodynamic Screening of Tachykinin NK2 Antagonists
저자
by
Tanaka, Takahiro
;
Matsumoto-Okano, Shiho
;
Inatomi, Nobuhiro
;
Fujioka, Yasushi
;
Kamiguchi, Hidenori
, et al.
소스
In
Journal of Pharmacological Sciences
2012 118(4):487-495
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7 . Academic Journal
Effect of molecular charges on renal uptake of 111In-DTPA-conjugated peptides
저자
by
Akizawa, Hiromichi
;
Arano, Yasushi
;
Mifune, Masaki
;
Iwado, Akimasa
;
Saito, Yutaka
, et al.
소스
In
Nuclear Medicine and Biology
October 2001 28(7):761-768
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7 . Academic Journal
Significance of 111In-DTPA chelate in renal radioactivity levels of 111In-DTPA-conjugated peptides
저자
by
Akizawa, Hiromichi
;
Arano, Yasushi
;
Mifune, Masaki
;
Iwado, Akimasa
;
Saito, Yutaka
, et al.
소스
In
Nuclear Medicine and Biology
2001 28(4):459-468
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