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1 . Academic Journal
Group 3 medulloblastoma transcriptional networks collapse under domain specific EP300/CBP inhibition
저자
by
Noha A. M. Shendy
;
Melissa Bikowitz
;
Logan H. Sigua
;
Yang Zhang
;
Audrey Mercier
, et al.
소스
Nature Communications, Vol 15, Iss 1, Pp 1-18 (2024)
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7 . Academic Journal
Development of allosteric and selective CDK2 inhibitors for contraception with negative cooperativity to cyclin binding
저자
by
Erik B. Faber
;
Luxin Sun
;
Jian Tang
;
Emily Roberts
;
Sornakala Ganeshkumar
, et al.
소스
Nature Communications, Vol 14, Iss 1, Pp 1-13 (2023)
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7 . Academic Journal
SARS-CoV-2 Period Seroprevalence and Related Factors, Hillsborough County, Florida, USA, October 2020–March 2021
저자
by
Anna R. Giuliano
;
Shari Pilon-Thomas
;
Michael J. Schell
;
Martha Abrahamsen
;
Jessica Y. Islam
, et al.
소스
Emerging Infectious Diseases, Vol 28, Iss 3, Pp 556-563 (2022)
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7 . Academic Journal
Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations
저자
by
Bryce K. Allen
;
Saurabh Mehta
;
Stuart W. J. Ember
;
Jin-Yi Zhu
;
Ernst Schönbrunn
, et al.
소스
ACS Omega, Vol 2, Iss 8, Pp 4760-4771 (2017)
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7 . Academic Journal
Stability of the Human Hsp90-p50Cdc37 Chaperone Complex against Nucleotides and Hsp90 Inhibitors, and the Influence of Phosphorylation by Casein Kinase 2
저자
by
Sanne H. Olesen
;
Donna J. Ingles
;
Jin-Yi Zhu
;
Mathew P. Martin
;
Stephane Betzi
, et al.
소스
Molecules, Vol 20, Iss 1, Pp 1643-1660 (2015)
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7 . Academic Journal
Ack1 mediated AKT/PKB tyrosine 176 phosphorylation regulates its activation.
저자
by
Kiran Mahajan
;
Domenico Coppola
;
Sridevi Challa
;
Bin Fang
;
Y Ann Chen
, et al.
소스
PLoS ONE, Vol 5, Iss 3, p e9646 (2010)
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7 .
Screening through Lead Optimization of High Affinity, Allosteric Cyclin-Dependent Kinase 2 (CDK2) Inhibitors as Male Contraceptives That Reduce Sperm Counts in Mice
저자
by
Erik B. Faber
;
Nan Wang
;
Kristen John
;
Luxin Sun
;
Henry L. Wong
, et al.
소스
Journal of Medicinal Chemistry
. 66:1928-1940
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7 .
Chemical Proteomics with Novel Fully Functionalized Fragments and Stringent Target Prioritization Identifies the Glutathione-Dependent Isomerase GSTZ1 as a Lung Cancer Target
저자
by
Yi Liao
;
Sean Chin Chan
;
Eric A. Welsh
;
Bin Fang
;
Luxin Sun
, et al.
소스
ACS Chemical Biology
. 18:251-264
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7 .
Bivalent BET Bromodomain Inhibitors Confer Increased Potency and Selectivity for BRDT via Protein Conformational Plasticity
저자
by
Xianghong Guan
;
Narsihmulu Cheryala
;
Rezaul Md. Karim
;
Alice Chan
;
Norbert Berndt
, et al.
소스
Journal of Medicinal Chemistry
. 65:10441-10458
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7 .
Supplementary Data from EP300 Selectively Controls the Enhancer Landscape of MYCN-Amplified Neuroblastoma
저자
by
Jun Qi
;
A. Thomas Look
;
Kimberly Stegmaier
;
Brian J. Abraham
;
Martha L. Bulyk
, et al.
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