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1 . Academic Journal
Preclinical alternative drug discovery programs for monogenic rare diseases. Should small molecules or gene therapy be used? The case of hereditary spastic paraplegias
저자
by
Caron, Giulia
;
Lamacchia, Lorenzo
;
Francisco, Serena
;
Brusco, Alfredo
;
Pullano, Verdiana
, et al.
소스
In
Drug Discovery Today
October 2024 29(10)
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7 . Academic Journal
Exploring the chemical space of orally bioavailable PROTACs
저자
by
Apprato, Giulia
;
Poongavanam, Vasanthanathan
;
Garcia Jimenez, Diego
;
Atilaw, Yoseph
;
Erdelyi, Mate
, et al.
소스
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Drug Discovery Today
April 2024 29(4)
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7 . Academic Journal
Ionization and lipophilicity in nonpolar media mimicking the cell membrane interior
저자
by
Vallaro, Maura
;
Ermondi, Giuseppe
;
Saame, Jaan
;
Leito, Ivo
;
Caron, Giulia
.
소스
In
Bioorganic & Medicinal Chemistry
1 March 2023 81
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7 . Academic Journal
Characterization of the new CelerisTM Arginine column: Retentive behaviour through a combination of chemometric tools and potential in drug analysis
저자
by
Russo, Giacomo
;
Vallaro, Maura
;
Cappelli, Luca
;
Anderson, Scott
;
Ermondi, Giuseppe
, et al.
소스
In
Journal of Chromatography A
16 August 2021 1651
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7 . Academic Journal
Predicting the Permeability of Macrocycles from Conformational Sampling – Limitations of Molecular Flexibility
저자
by
Poongavanam, Vasanthanathan
;
Atilaw, Yoseph
;
Ye, Sofie
;
Wieske, Lianne H.E.
;
Erdelyi, Mate
, et al.
소스
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Journal of Pharmaceutical Sciences
January 2021 110(1):301-313
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7 . Academic Journal
Degraders early developability assessment: face-to-face with molecular properties
저자
by
Ermondi, Giuseppe
;
Vallaro, Maura
;
Caron, Giulia
.
소스
In
Drug Discovery Today
September 2020 25(9):1585-1591
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5 . Academic Journal
Flexibility in early drug discovery: focus on the beyond-Rule-of-5 chemical space
저자
by
Caron, Giulia
;
Digiesi, Vito
;
Solaro, Sara
;
Ermondi, Giuseppe
.
소스
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Drug Discovery Today
April 2020 25(4):621-627
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6 . Academic Journal
IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs.
저자
by
Garcia Jimenez, Diego
;
Rossi Sebastiano, Matteo
;
Vallaro, Maura
;
Ermondi, Giuseppe
;
Caron, Giulia
.
소스
Journal of Medicinal Chemistry; 7/11/2024, Vol. 67 Issue 13, p11421-11434, 14p
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7 . Academic Journal
Log P as a tool in intramolecular hydrogen bond considerations
저자
by
Caron, Giulia
;
Vallaro, Maura
;
Ermondi, Giuseppe
.
소스
In
Drug Discovery Today: Technologies
July 2018 27:65-70
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5 . Academic Journal
Learning how to use IAM chromatography for predicting permeability
저자
by
Ermondi, Giuseppe
;
Vallaro, Maura
;
Caron, Giulia
.
소스
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European Journal of Pharmaceutical Sciences
1 March 2018 114:385-390
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