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1 . Academic Journal
Discovery and X-ray Crystallographic Analysis of a Spiropiperidine Iminohydantoin Inhibitor of β-Secretase.
저자
by
James C. Barrow
;
Shaun R. Stauffer
;
Kenneth E. Rittle
;
Phung L. Ngo
;
ZhiQiang Yang
, et al.
소스
Journal of Medicinal Chemistry
. Oct2008, Vol. 51 Issue 20, p6259-6262. 4p.
Full Text (ACS)
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7 .
Development of a pharmacodynamic biomarker to measure target engagement from inhibition of the NGF–TrkA pathway
저자
by
Shawn J. Stachel
;
Kausik K. Nanda
;
Darrell A. Henze
;
Eric A. Price
;
Alicja Krasowska-Zoladek
.
소스
Journal of Neuroscience Methods
. 282:34-42
Web of Science
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7 . Academic Journal
Discovery of Isonicotinamide Derived -Secretase Inhibitors: In Vivo Reduction of -Amyloid.
저자
by
Matthew G. Stanton
;
Shaun R. Stauffer
;
Alison R. Gregro
;
Melissa Steinbeiser
;
Philippe Nantermet
, et al.
소스
Journal of Medicinal Chemistry
. Jul2007, Vol. 50 Issue 15, p3431-3433. 3p.
Full Text (ACS)
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7 .
Cisterna magna cannulated repeated CSF sampling rat model – effects of a gamma-secretase inhibitor on Aβ levels
저자
by
Eric A. Price
;
Adam J. Simon
;
Jennifer S. Shapiro
;
Sethu Sankaranarayanan
;
Mark Stiteler
, et al.
소스
Journal of Neuroscience Methods
. 205:36-44
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7 .
Acute γ-Secretase Inhibition of Nonhuman Primate CNS Shifts Amyloid Precursor Protein (APP) Metabolism from Amyloid-β Production to Alternative APP Fragments without Amyloid-β Rebound
저자
by
Eric A. Price
;
Gene G. Kinney
;
Randall J. Bateman
;
Maria S. Michener
;
Marie A. Holahan
, et al.
소스
The Journal of Neuroscience
. 30:6743-6750
Open Access (OpenAIRE)
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7 .
First Demonstration of Cerebrospinal Fluid and Plasma Aβ Lowering with Oral Administration of a β-Site Amyloid Precursor Protein-Cleaving Enzyme 1 Inhibitor in Nonhuman Primates
저자
by
Janet Lineberger
;
Matthew G. Stanton
;
Amy S. Espeseth
;
Beth Pietrak
;
Min Xu
, et al.
소스
Journal of Pharmacology and Experimental Therapeutics
. 328:131-140
Web of Science
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7 .
Discovery and X-ray Crystallographic Analysis of a Spiropiperidine Iminohydantoin Inhibitor of β-Secretase
저자
by
Kenneth E. Rittle
;
Dorothy Levorse
;
James C. Barrow
;
Eric A. Price
;
Katherine Tugusheva
, et al.
소스
Journal of Medicinal Chemistry
. 51:6259-6262
Web of Science
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7 .
In Vivo β-Secretase 1 Inhibition Leads to Brain Aβ Lowering and Increased α-Secretase Processing of Amyloid Precursor Protein without Effect on Neuregulin-1
저자
by
Guoxin Wu
;
Craig A. Coburn
;
Lixia Jin
;
Joan D. Ellis
;
Adam J. Simon
, et al.
소스
Journal of Pharmacology and Experimental Therapeutics
. 324:957-969
Web of Science
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7 .
Nanometer Distance Measurements in RNA Using Site-Directed Spin Labeling
저자
by
Kálmán Hideg
;
Eric A. Price
;
Peter Z. Qin
;
Qi Cai
;
Ian S. Haworth
, et al.
소스
Biophysical Journal
. 93(6):2110-2117
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7 .
Compounds That Bind APP and Inhibit Aβ Processing in Vitro Suggest a Novel Approach to Alzheimer Disease Therapeutics
저자
by
Elizabeth Chen Dodson
;
Janet Lineberger
;
Adam J. Simon
;
Ming-Tain Lai
;
Mohinder K. Sardana
, et al.
소스
Journal of Biological Chemistry
. 280:17792-17797
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