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1 . Academic Journal
Case Studies of Minimizing Nonspecific Inhibitors in HTS Campaigns That Use Assay-Ready Plates
저자
by
Liu, Yichin
;
Beresini, Maureen H.
;
Johnson, Adam
;
Mintzer, Robert
;
Shah, Kinjalkumar
, et al.
소스
In
SLAS Discovery
February 2012 17(2):225-236
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7 . Academic Journal
Antagonists of inhibitor of apoptosis proteins based on thiazole amide isosteres
저자
by
Cohen, Frederick
;
Koehler, Michael F.T.
;
Bergeron, Philippe
;
Elliott, Linda O.
;
Flygare, John A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(7):2229-2233
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7 . Academic Journal
Erratum to “Antagonists of inhibitor of apoptosis proteins based on thiazole amide isosteres” [Bioorg. Med. Chem. Lett. 20 (2010) 2229–2233]
저자
by
Cohen, Frederick
;
Koehler, Michael F.T.
;
Bergeron, Philippe
;
Elliott, Linda O.
;
Flygare, John A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 January 2012 22(1):753-754
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7 . Academic Journal
Discovery of a PotentSmall-Molecule Antagonist of Inhibitor of Apoptosis (IAP) Proteins andClinical Candidate for the Treatment of Cancer (GDC-0152).
저자
by
Flygare, John A.
;
Beresini, Maureen
;
Budha, Nageshwar
;
Chan, Helen
;
Chan, Iris T.
, et al.
소스
Journal of Medicinal Chemistry
. May2012, Vol. 55 Issue 9, p4101-4113. 13p.
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7 . Academic Journal
IAP Antagonists Induce Autoubiquitination of c-IAPs, NF-κB Activation, and TNFα-Dependent Apoptosis
저자
by
Varfolomeev, Eugene
;
Blankenship, John W.
;
Wayson, Sarah M.
;
Fedorova, Anna V.
;
Kayagaki, Nobuhiko
, et al.
소스
Cell
. Nov2007, Vol. 131 Issue 4, p669-681. 13p.
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7 . Academic Journal
A Selective, Slow Binding Inhibitor of Factor VIIa Binds to a Nonstandard Active Site Conformation and Attenuates Thrombus Formation in Vivo.
저자
by
Olivero, Alan G.
;
Eigenbrot, Charles
;
Goldsmith, Richard
;
Robarge, Kirk
;
Artis, Dean R.
, et al.
소스
Journal of Biological Chemistry
. 3/11/2005, Vol. 280 Issue 10, p9160-9169. 10p. 5 Diagrams, 5 Charts, 4 Graphs.
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7 . Academic Journal
Structure and Function Analysis of Peptide Antagonists of Melanoma Inhibitor of Apoptosis (ML-IAP).
저자
by
Franklin, Matthew C.
;
Kadkhodayan, Saloumeh
;
Ackerly, Heidi
;
Alexandru, Daniela
;
Distefano, Mark D.
, et al.
소스
Biochemistry
. 7/15/2003, Vol. 42 Issue 27, p8223. 9p. 5 Diagrams, 2 Charts, 3 Graphs.
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7 . Periodical
Antagonism of c-IAP and XIAP Proteins Is Required for Efficient Induction of Cell Death by Small-Molecule IAP Antagonists
저자
by
Ndubaku, Chudi
;
Varfolomeev, Eugene
;
Wang, Lan
;
Zobel, Kerry
;
Lau, Kevin
, et al.
소스
ACS Chemical Biology; July 2009, Vol. 4 Issue: 7 p557-566, 10p
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7 . Periodical
Design, Synthesis, and Biological Activity of a Potent Smac Mimetic That Sensitizes Cancer Cells to Apoptosis by Antagonizing IAPs
저자
by
Zobel, Kerry
;
Wang, Lan
;
Varfolomeev, Eugene
;
Franklin, Matthew C.
;
Elliott, Linda O.
, et al.
소스
ACS Chemical Biology; September 2006, Vol. 1 Issue: 8 p525-533, 9p
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7 . Periodical
Engineering ML-IAP to produce an extraordinarily potent caspase 9 inhibitor: implications for Smac-dependent anti-apoptotic activity of ML-IAP
저자
by
VUCIC, Domagoj
;
FRANKLIN, Matthew C.
;
WALLWEBER, Heidi J. A.
;
DAS, Kanad
;
ECKELMAN, Brendan P.
, et al.
소스
Biochemical Journal; January 2005, Vol. 385 Issue: 1 p11-20, 10p
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