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1 . Academic Journal
Design, synthesis, and anti-proliferative evaluation of new quinazolin-4(3H)-ones as potential VEGFR-2 inhibitors
저자
by
El-Adl, Khaled
;
El-Helby, Abdel-Ghany A.
;
Ayyad, Rezk R.
;
Mahdy, Hazem A.
;
Khalifa, Mohamed M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 January 2021 29
Full Text (ScienceDirect)
Scopus
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7 . Academic Journal
Triazoloquinoxalines-based DNA intercalators-Topo II inhibitors: design, synthesis, docking, ADMET and anti-proliferative evaluations.
저자
by
Elwan, Alaa
;
Sakr, Helmy
;
El-Helby, Abdel-Ghany A.
;
El-morsy, Ahmed
;
Abdelgawad, Mohamed A.
, et al.
소스
Journal of Enzyme Inhibition & Medicinal Chemistry
. 2022, Vol. 37 Issue 1, p1556-1567. 12p.
Open Access (T&F)
Scopus
Web of Science
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7 . Academic Journal
Design, synthesis, docking, ADMET profile, and anticancer evaluations of novel thiazolidine‐2,4‐dione derivatives as VEGFR‐2 inhibitors.
저자
by
El‐Adl, Khaled
;
Sakr, Helmy
;
El‐Hddad, Sanadelaslam S. A.
;
El‐Helby, Abdel‐Ghany A.
;
Nasser, Mohamed
, et al.
소스
Archiv der Pharmazie; Jul2021, Vol. 354 Issue 7, p1-18, 18p
Scopus
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7 . Academic Journal
Design, synthesis, molecular docking, anticancer evaluations, and in silico pharmacokinetic studies of novel 5‐[(4‐chloro/2,4‐dichloro)benzylidene]thiazolidine‐2,4‐dione derivatives as VEGFR‐2 inhibitors.
저자
by
El‐Adl, Khaled
;
El‐Helby, Abdel‐Ghany A.
;
Sakr, Helmy
;
Ayyad, Rezk R.
;
Mahdy, Hazem A.
, et al.
소스
Archiv der Pharmazie; Feb2021, Vol. 354 Issue 2, p1-17, 17p
Scopus
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7 . Academic Journal
[1,2,4]Triazolo[4,3-a]quinoxaline and [1,2,4]triazolo[4,3-a]quinoxaline-1-thiol-derived DNA intercalators: design, synthesis, molecular docking, in silico ADMET profiles and anti-proliferative evaluations.
저자
by
El-Adl, Khaled
;
El-Helby, Abdel-Ghany A.
;
Sakr, Helmy
;
Elwan, Alaa
.
소스
New Journal of Chemistry
. 1/14/2021, Vol. 45 Issue 2, p881-897. 17p.
Full Text (RSC Gold)
Scopus
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6 . Academic Journal
Design, synthesis, molecular docking, and anticancer evaluations of 1‐benzylquinazoline‐2,4(1H,3H)‐dione bearing different moieties as VEGFR‐2 inhibitors.
저자
by
El‐Adl, Khaled
;
El‐Helby, Abdel‐Ghany A.
;
Sakr, Helmy
;
El‐Hddad, Sanadelaslam S. A.
.
소스
Archiv der Pharmazie; Aug2020, Vol. 353 Issue 8, p1-14, 14p
Scopus
Web of Science
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6 . Academic Journal
Phthalazine-1,4-dione derivatives as non-competitive AMPA receptor antagonists: design, synthesis, anticonvulsant evaluation, ADMET profile and molecular docking.
저자
by
El-Helby, Abdel-Ghany A.
;
Ayyad, Rezk R. A.
;
El-Adl, Khaled
;
Elkady, Hazem
.
소스
Molecular Diversity; May2019, Vol. 23 Issue 2, p283-298, 16p
Scopus
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6 . Periodical
Design, Synthesis, In VitroAnti-cancer Activity, ADMET Profile and Molecular Docking of Novel Triazolo[3,4-a]phthalazine Derivatives Targeting VEGFR-2 Enzyme
저자
by
El-Helby, Abdel-Ghany A.
;
Sakr, Helmy
;
Ayyad, Rezk R.A.
;
El-Adl, Khaled
;
Ali, Mamdouh M.
, et al.
소스
Anti-Cancer Agents in Medicinal Chemistry; June 2018, Vol. 18 Issue: 8 p1184-1196, 13p
Full Text (Bentham Science)
Scopus
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7 . Academic Journal
Discovery of new quinazolin-4(3H)-ones as VEGFR-2 inhibitors: Design, synthesis, and anti-proliferative evaluation
저자
by
Eissa, Ibrahim H.
;
El-Helby, Abdel-Ghany A.
;
Mahdy, Hazem A.
;
Khalifa, Mohamed M.
;
Elnagar, Hamdy A.
, et al.
소스
BIOORGANIC CHEMISTRY
; DEC 2020, 105 p104380 13p.
Full Text (ScienceDirect)
Scopus
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7 . Academic Journal
Design, synthesis, molecular docking and anti-proliferative evaluations of [1,2,4]triazolo[4,3-a]quinoxaline derivatives as DNA intercalators and Topoisomerase II inhibitors
저자
by
El-Adl, Khaled
;
El-Helby, Abdel-Ghany A.
;
Sakr, Helmy
;
Elwan, Alaa
.
소스
BIOORGANIC CHEMISTRY
; DEC 2020, 105 p104399 19p.
Full Text (ScienceDirect)
Scopus
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