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1 . Academic Journal
Modulation of taxane binding to tubulin curved and straight conformations by systematic 3′N modification provides for improved microtubule binding, persistent cytotoxicity and in vivo potency
저자
by
Ma, Yuntao
;
Josa-Prado, Fernando
;
Essif, Jacob Nathaniel
;
Liu, Shuqi
;
Li, Shuo
, et al.
소스
In
European Journal of Medicinal Chemistry
5 November 2023 259
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7 . Academic Journal
Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy
저자
by
Campiani, Giuseppe
;
Khan, Tuhina
;
Ulivieri, Cristina
;
Staiano, Leopoldo
;
Papulino, Chiara
, et al.
소스
In
European Journal of Medicinal Chemistry
5 May 2022 235
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7 . Academic Journal
Diphenyl ether derivatives occupy the expanded binding site of cyclohexanedione compounds at the colchicine site in tubulin by movement of the αT5 loop
저자
by
Bueno, Oskia
;
Gargantilla, Marta
;
Estévez-Gallego, Juan
;
Martins, Solange
;
Díaz, J. Fernando
, et al.
소스
In
European Journal of Medicinal Chemistry
1 June 2019 171:195-208
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7 . Academic Journal
Structure-activity relationships, biological evaluation and structural studies of novel pyrrolonaphthoxazepines as antitumor agents
저자
by
Brindisi, Margherita
;
Ulivieri, Cristina
;
Alfano, Gloria
;
Gemma, Sandra
;
de Asís Balaguer, Francisco
, et al.
소스
In
European Journal of Medicinal Chemistry
15 January 2019 162:290-320
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7 . Academic Journal
Modification of C-seco taxoids through ring tethering and substituent replacement leading to effective agents against tumor drug resistance mediated by βIII-Tubulin and P-glycoprotein (P-gp) overexpressions
저자
by
Tang, Yong
;
Rodríguez-Salarichs, Javier
;
Zhao, Yu
;
Cai, Pei
;
Estévez-Gallego, Juan
, et al.
소스
In
European Journal of Medicinal Chemistry
8 September 2017 137:488-503
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7 . Academic Journal
Development of Potent Microtubule Targeting Agent by Structural Simplification of Natural Diazonamide.
저자
by
Kalnins, Toms
;
Vitkovska, Viktorija
;
Kazak, Mihail
;
Zelencova-Gopejenko, Diana
;
Ozola, Melita
, et al.
소스
Journal of Medicinal Chemistry; 6/13/2024, Vol. 67 Issue 11, p9227-9259, 33p
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7 . Academic Journal
High affinity and covalent-binding microtubule stabilizing agents show activity in chemotherapy-resistant acute myeloid leukemia cells
저자
by
Pera, Benet
;
Calvo-Vidal, M. Nieves
;
Ambati, Srikanth
;
Jordi, Michel
;
Kahn, Alissa
, et al.
소스
In
Cancer Letters
1 November 2015 368(1):97-104
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7 . Academic Journal
PM534, an Optimized Target-Protein Interaction Strategy through the Colchicine Site of Tubulin.
저자
by
Lucena-Agell, Daniel
;
Guillén, María José
;
Matesanz, Ruth
;
Álvarez-Bernad, Beatriz
;
Hortigüela, Rafael
, et al.
소스
Journal of Medicinal Chemistry; 2/22/2024, Vol. 678 Issue 4, p2619-2630, 12p
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7 . Academic Journal
Taxanes with high potency inducing tubulin assembly overcome tumoural cell resistances
저자
by
Matesanz, Ruth
;
Trigili, Chiara
;
Rodríguez-Salarichs, Javier
;
Zanardi, Ilaria
;
Pera, Benet
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 September 2014 22(18):5078-5090
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7 . Academic Journal
Tannic Acid and Ethyl Gallate Potentialize Paclitaxel Effect on Microtubule Dynamics in Hep3B Cells.
저자
by
Sánchez-Carranza, Jessica Nayelli
;
Redondo-Horcajo, Mariano
;
Barasoain, Isabel
;
Escobar-Aguilar, Ever Angel
;
Millán-Pacheco, César
, et al.
소스
Pharmaceuticals (14248247)
. Nov2023, Vol. 16 Issue 11, p1579. 20p.
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