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1 . Academic Journal
Selective inhibition of indoleamine and tryptophan 2,3-dioxygenases: Comparative study on kynurenine pathway in cell lines via LC-MS/MS-based targeted metabolomics
저자
by
Villani, Salvatore
;
Fallarini, Silvia
;
Rezzi, Sarah Jane
;
Di Martino, Rita Maria Concetta
;
Aprile, Silvio
, et al.
소스
In
Journal of Pharmaceutical and Biomedical Analysis
5 January 2024 237
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7 . Academic Journal
Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffold
저자
by
De Lorenzi, Ersilia
;
Seghetti, Francesca
;
Tarozzi, Andrea
;
Pruccoli, Letizia
;
Contardi, Cecilia
, et al.
소스
In
European Journal of Medicinal Chemistry
5 April 2023 252
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7 . Academic Journal
Novel fragment-derived colchicine-site binders as microtubule-destabilizing agents
저자
by
de la Roche, Noelia Montel
;
Mühlethaler, Tobias
;
Di Martino, Rita Maria Concetta
;
Ortega, Jose Antonio
;
Gioia, Dario
, et al.
소스
In
European Journal of Medicinal Chemistry
5 November 2022 241
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7 . Periodical
Deuterium in drug discovery: progress, opportunities and challenges
저자
by
Di Martino, Rita Maria Concetta
;
Maxwell, Brad D.
;
Pirali, Tracey
.
소스
Nature Reviews Drug Discovery; July 2023, Vol. 22 Issue: 7 p562-584, 23p
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5 . Academic Journal
A Versatile and Sustainable Multicomponent Platform for the Synthesis of Protein Degraders: Proof-of-Concept Application to BRD4-Degrading PROTACs.
저자
by
Bhela, Irene Preet
;
Ranza, Alice
;
Balestrero, Federica Carolina
;
Serafini, Marta
;
Aprile, Silvio
, et al.
소스
Journal of Medicinal Chemistry; 11/24/2022, Vol. 65 Issue 22, p15282-15299, 18p
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7 . Academic Journal
Modulation of Amyloid β-Induced Microglia Activation and Neuronal Cell Death by Curcumin and Analogues.
저자
by
De Lorenzi, Ersilia
;
Franceschini, Davide
;
Contardi, Cecilia
;
Di Martino, Rita Maria Concetta
;
Seghetti, Francesca
, et al.
소스
International Journal of Molecular Sciences
. Apr2022, Vol. 23 Issue 8, p4381-4381. 21p.
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7 . Periodical
Dopamine D3 receptor ligands: a patent review (2014–2020)
저자
by
Di Martino, Rita Maria Concetta
;
Cavalli, Andrea
;
Bottegoni, Giovanni
.
소스
Expert Opinion on Therapeutic Patents; June 2022, Vol. 32 Issue: 6 p605-627, 23p
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5 . Academic Journal
From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold
저자
by
Rampa, Angela
;
Mancini, Francesca
;
De Simone, Angela
;
Falchi, Federico
;
Belluti, Federica
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 July 2015 25(14):2804-2808
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7 . Academic Journal
Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease.
저자
by
Di Martino, Rita Maria Concetta
;
Pruccoli, Letizia
;
Bisi, Alessandra
;
Gobbi, Silvia
;
Rampa, Angela
, et al.
소스
ACS Chemical Neuroscience; 9/2/2020, Vol. 11 Issue 17, p2728-2740, 13p
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7 . Academic Journal
Multitarget Compounds for Bipolar Disorder: From Rational Design to Preliminary Pharmacokinetic Evaluation.
저자
by
Di Martino, Rita Maria Concetta
;
Bottegoni, Giovanni
;
Seghetti, Francesca
;
Russo, Debora
;
Penna, Ilaria
, et al.
소스
ChemMedChem; 6/4/2020, Vol. 15 Issue 11, p949-954, 6p
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