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1 . Academic Journal
Synthesis and structure activity relationship of the first class of LXR inverse agonists
저자
by
Elgendy, Bahaa
;
Griffett, Kristine
;
Hegazy, Lamees
;
Di Fruscia, Paolo
;
Sample, Kirby
, et al.
소스
In
Bioorganic Chemistry
February 2022 119
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7 . Academic Journal
Discovery of 5-{4-[(7-Ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-3-yl)methyl]piperazin-1-yl}-N-methyl-pyridine-2-carboxamide (AZD5305): A PARP1-DNA Trapper with High Selectivity for PARP1 over PARP2 and Other PARPs.
저자
by
Johannes, Jeffrey W.
;
Balazs, Amber
;
Barratt, Derek
;
Bista, Michal
;
Chuba, Matthew D.
, et al.
소스
Journal of Medicinal Chemistry; 10/14/2021, Vol. 64 Issue 19, p14498-14512, 15p
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7 . Academic Journal
The discovery of indole full agonists of the neurotensin receptor 1 (NTSR1)
저자
by
Di Fruscia, Paolo
;
He, Yuanjun
;
Koenig, Marcel
;
Tabrizifard, Sahba
;
Nieto, Ainhoa
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 August 2014 24(16):3974-3978
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7 . Periodical
Discovery of 5-{4-[(7-Ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-3-yl)methyl]piperazin-1-yl}-N-methylpyridine-2-carboxamide (AZD5305): A PARP1–DNA Trapper with High Selectivity for PARP1 over PARP2 and Other PARPs
저자
by
Johannes, Jeffrey W.
;
Balazs, Amber
;
Barratt, Derek
;
Bista, Michal
;
Chuba, Matthew D.
, et al.
소스
Journal of Medicinal Chemistry; October 2021, Vol. 64 Issue: 19 p14498-14512, 15p
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7 . Academic Journal
Fragment-Based Discovery of Novel Allosteric MEK1 Binders.
저자
by
Di Fruscia, Paolo
;
Edfeldt, Fredrik
;
Shamovsky, Igor
;
Collie, Gavin W.
;
Aagaard, Anna
, et al.
소스
ACS Medicinal Chemistry Letters; 2/11/2021, Vol. 12 Issue 2, p302-308, 7p
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7 . Academic Journal
Identification, Structure–Activity Relationship, and Biological Characterization of 2,3,4,5-Tetrahydro‑1H‑pyrido[4,3‑b]indoles as a Novel Class of CFTR Potentiators.
저자
by
Brindani, Nicoletta
;
Gianotti, Ambra
;
Giovani, Simone
;
Giacomina, Francesca
;
Di Fruscia, Paolo
, et al.
소스
Journal of Medicinal Chemistry; 10/8/2020, Vol. 63 Issue 19, p11169-11194, 26p
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7 . Dissertation/ Thesis
The design, synthesis and biological evaluation of novel small-molecule HDAC inhibitors
저자
by
Di Fruscia, Paolo
;
Fuchter, Matthew
;
Stronach, Euan
.
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5 . Periodical
Put a ring on it: application of small aliphatic rings in medicinal chemistryAll authors contributed to writing the manuscript.
저자
by
Bauer, Matthias R.
;
Di Fruscia, Paolo
;
Lucas, Simon C. C.
;
Michaelides, Iacovos N.
;
Nelson, Jennifer E.
, et al.
소스
MedChemComm; 2021, Vol. 12 Issue: 4 p448-471, 24p
Find it @ DONGA
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7 .
Identification, Structure–Activity Relationship, and Biological Characterization of 2,3,4,5-Tetrahydro-1H-pyrido[4,3-b]indoles as a Novel Class of CFTR Potentiators
저자
by
Federico Sorana
;
Rosalia Bertorelli
;
Simone Giovani
;
Tiziano Bandiera
;
Giuliana Ottonello
, et al.
소스
Journal of Medicinal Chemistry
Open Access (OpenAIRE)
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7 . Academic Journal
Thienopyrimidinone Based Sirtuin-2 (SIRT2)-Selective Inhibitors Bind in the Ligand Induced Selectivity Pocket.
저자
by
Sundriyal, Sandeep
;
Moniot, Sébastien
;
Mahmud, Zimam
;
Shang Yao
;
Di Fruscia, Paolo
, et al.
소스
Journal of Medicinal Chemistry
. 3/9/2017, Vol. 60 Issue 5, p1928-1945. 18p.
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