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1 . Academic Journal
10-(2-Benzoxazolcarbonyl)-5,10-dideaza-acyclic-5,6,7,8-tetrahydrofolic acid: A potential inhibitor of GAR transformylase and AICAR transformylase
저자
by
Marsilje, Thomas H
;
Hedrick, Michael P
;
Desharnais, Joel
;
Capps, Kevin
;
Tavassoli, Ali
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2003 11(20):4503-4509
Full Text (ScienceDirect)
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7 . Academic Journal
Design, synthesis, and biological evaluation of simplified α-Keto heterocycle, trifluoromethyl ketone, and formyl substituted folate analogues as potential inhibitors of GAR transformylase and AICAR transformylase
저자
by
Marsilje, Thomas H
;
Hedrick, Michael P
;
Desharnais, Joel
;
Tavassoli, Ali
;
Zhang, Yan
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2003 11(20):4487-4501
Full Text (ScienceDirect)
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7 . Academic Journal
Design, synthesis and biological evaluation of 10-CF 3CO-DDACTHF analogues and derivatives as inhibitors of GAR Tfase and the de novo purine biosynthetic pathway
저자
by
Desharnais, Joel
;
Hwang, Inkyu
;
Zhang, Yan
;
Tavassoli, Ali
;
Baboval, Justin
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2003 11(20):4511-4521
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7 . Academic Journal
10-Formyl-5,10-dideaza-acyclic-5,6,7,8-tetrahydrofolic acid (10-Formyl-DDACTHF): A potent cytotoxic agent acting by selective inhibition of human GAR Tfase and the de novo purine biosynthetic pathway
저자
by
Marsilje, Thomas H.
;
Labroli, Marc A.
;
Hedrick, Michael P.
;
Jin, Qing
;
Desharnais, Joel
, et al.
소스
In
Bioorganic & Medicinal Chemistry
August 2002 10(8):2739-2749
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7 . Academic Journal
Kinase-mediated trapping of bi-functional conjugates of paclitaxel or vinblastine with thymidine in cancer cells
저자
by
Aspland, Simon E.
;
Ballatore, Carlo
;
Castillo, Rosario
;
Desharnais, Joel
;
Eustaquio, Trisha
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2006 16(19):5194-5198
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7 . Academic Journal
A facile route to paclitaxel C-10 carbamates
저자
by
Ballatore, Carlo
;
Aspland, Simon E.
;
Castillo, Rosario
;
Desharnais, Joel
;
Eustaquio, Trisha
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
16 May 2005 15(10):2477-2480
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7 . Academic Journal
Pyroglutamate and O-Linked Glycan Determine Functional Production of Anti-IL17A and Anti-IL22 Peptide-Antibody Bispecific Genetic Fusions.
저자
by
Xiaotian Zhong
;
Kieras, Elizabeth
;
Sousa, Eric
;
D'Antona, Aaron
;
Baber, J. Christian
, et al.
소스
Journal of Biological Chemistry
. 1/11/2013, Vol. 288 Issue 2, p1409-1419. 11p.
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7 . Academic Journal
Design, synthesis and biological evaluation of 10-CF
3
CO-DDACTHF analogues and derivatives as inhibitors of GAR Tfase and the de novo purine biosynthetic pathway
저자
by
Desharnais, Joel
;
Hwang, Inkyu
;
Zhang, Yan
;
Tavassoli, Ali
;
Baboval, Justin
, et al.
소스
Bioorganic & Medicinal Chemistry
. Oct2003, Vol. 11 Issue 20, p4511. 11p.
Full Text (ScienceDirect)
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7 . Academic Journal
Rational Design, Synthesis, Evaluation, and Crystal Structure of a Potent Inhibitor of Human GAR Tfase: 10-(Trifluoroacetyl)-5, 10-dideazaacyclic-5,6,7,8-tetrahydrofolic Acid.
저자
by
Yan Zhang
;
Desharnais, Joel
;
Marsilje, Thomas H.
;
Chenglong Li
;
Hedrick, Michael P.
, et al.
소스
Biochemistry
. 5/27/2003, Vol. 42 Issue 20, p6043. 14p. 20 Diagrams, 5 Charts.
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7 . Academic Journal
Crystal Structures of Human GAR Tfase at Low and High pH and with Substrate β-GAR.
저자
by
Yan Zhang
;
Desharnais, Joel
;
Greasley, Samantha E.
;
Beardsley, G. Peter
;
Boger, Dale L.
, et al.
소스
Biochemistry
. 12/3/2002, Vol. 41 Issue 48, p14206. 10p. 14 Diagrams, 1 Chart, 1 Graph.
Full Text (ACS)
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