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1 . Academic Journal
Discovery and X-ray Crystallographic Analysis of a Spiropiperidine Iminohydantoin Inhibitor of β-Secretase.
저자
by
James C. Barrow
;
Shaun R. Stauffer
;
Kenneth E. Rittle
;
Phung L. Ngo
;
ZhiQiang Yang
, et al.
소스
Journal of Medicinal Chemistry
. Oct2008, Vol. 51 Issue 20, p6259-6262. 4p.
Full Text (ACS)
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7 . Academic Journal
Discovery of Isonicotinamide Derived -Secretase Inhibitors: In Vivo Reduction of -Amyloid.
저자
by
Matthew G. Stanton
;
Shaun R. Stauffer
;
Alison R. Gregro
;
Melissa Steinbeiser
;
Philippe Nantermet
, et al.
소스
Journal of Medicinal Chemistry
. Jul2007, Vol. 50 Issue 15, p3431-3433. 3p.
Full Text (ACS)
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7 .
Discovery of pyrrolidine-based β-secretase inhibitors: Lead advancement through conformational design for maintenance of ligand binding efficiency
저자
by
Georgia B. McGaughey
;
Samuel L. Graham
;
M. Katharine Holloway
;
Sharie J. Haugabook
;
Paul Zuck
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 22:240-244
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7 .
Discovery of aminoheterocycles as a novel β-secretase inhibitor class: pH dependence on binding activity part 1
저자
by
Beth Pietrak
;
Hemaka A. Rajapakse
;
Dennis Colussi
;
Paul Zuck
;
Hong Zhu
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 19:2977-2980
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7 .
Evolution of Tertiary Carbinamine BACE‐1 Inhibitors: Aβ Reduction in Rhesus CSF upon Oral Dosing
저자
by
John Swestock
;
Ming Tain Lai
;
Shaun R. Stauffer
;
Sanjeev Munshi
;
Georgia B. McGaughey
, et al.
소스
ChemMedChem
. 4:37-40
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7 .
Identification of a small molecule β-secretase inhibitor that binds without catalytic aspartate engagement
저자
by
Amy S. Espeseth
;
Ivory D. Hills
;
Shawn J. Stachel
;
Thomas G. Steele
;
Georgia B. McGaughey
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 19:17-20
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7 .
First Demonstration of Cerebrospinal Fluid and Plasma Aβ Lowering with Oral Administration of a β-Site Amyloid Precursor Protein-Cleaving Enzyme 1 Inhibitor in Nonhuman Primates
저자
by
Janet Lineberger
;
Matthew G. Stanton
;
Amy S. Espeseth
;
Beth Pietrak
;
Min Xu
, et al.
소스
Journal of Pharmacology and Experimental Therapeutics
. 328:131-140
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7 .
Discovery and X-ray Crystallographic Analysis of a Spiropiperidine Iminohydantoin Inhibitor of β-Secretase
저자
by
Kenneth E. Rittle
;
Dorothy Levorse
;
James C. Barrow
;
Eric A. Price
;
Katherine Tugusheva
, et al.
소스
Journal of Medicinal Chemistry
. 51:6259-6262
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7 .
Design and Synthesis of 2,3,5-Substituted Imidazolidin-4-one Inhibitors of BACE-1
저자
by
Samuel L. Graham
;
Amy S. Espeseth
;
Kenneth E. Rittle
;
Katherine Tugusheva
;
Dennis Colussi
, et al.
소스
ChemMedChem
. 2:995-999
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7 .
β-Secretase (BACE-1) inhibitors: Accounting for 10s loop flexibility using rigid active sites
저자
by
Georgia B. McGaughey
;
Ming-Tain Lai
;
Hemaka A. Rajapakse
;
Sanjeev Munshi
;
Beth Pietrak
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 17:1117-1121
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