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1 . Academic Journal
Pharmacological characterization of RWJ-676070, a dual vasopressin V 1A/V 2 receptor antagonist
저자
by
Gunnet, Joseph W.
;
Wines, Pamela
;
Xiang, Min
;
Rybczynski, Philip
;
Andrade-Gordon, Patricia
, et al.
소스
In
European Journal of Pharmacology
2008 590(1):333-342
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7 . Academic Journal
Synthesis and biological evaluation of novel macrocyclic bis-7-azaindolylmaleimides as potent and highly selective glycogen synthase kinase-3β (GSK-3β) inhibitors
저자
by
Shen, Lan
;
Prouty, Catherine
;
Conway, Bruce R.
;
Westover, Lori
;
Xu, Jun Z.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 March 2004 12(5):1239-1255
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7 . Academic Journal
Design, synthesis, and biological evaluation of novel 7-azaindolyl-heteroaryl-maleimides as potent and selective glycogen synthase kinase-3β (GSK-3β) inhibitors
저자
by
O'Neill, David J.
;
Shen, Lan
;
Prouty, Catherine
;
Conway, Bruce R.
;
Westover, Lori
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2004 12(12):3167-3185
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7 . Academic Journal
A Branched DNA Signal Amplification Assay to Quantitate Messenger RNA of Human Uncoupling Proteins 1, 2, and 3
저자
by
Zhou, Lubing
;
Cryan, Ellen V.
;
Minor, Lisa K.
;
Gunnet, Joseph W.
;
Demarest, Keith T.
.
소스
In
Analytical Biochemistry
15 June 2000 282(1):46-53
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7 . Academic Journal
4-Bicyclic heteroaryl-piperidine derivatives as potent, orally bioavailable stearoyl-CoA desaturase-1 (SCD1) inhibitors: Part 2. Pyridazine-based analogs
저자
by
Yang, Shyh-Ming
;
Tang, Yuting
;
Rano, Thomas
;
Lu, Huajun
;
Kuo, Gee-Hong
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 March 2014 24(5):1437-1441
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7 . Academic Journal
4-Bicyclic heteroaryl-piperidine derivatives as potent, orally bioavailable Stearoyl-CoA desaturase-1 (SCD1) inhibitors. Part 1: Urea-based analogs
저자
by
Yang, Shyh-Ming
;
Tang, Yuting
;
Zhang, Rui
;
Lu, Huajun
;
Kuo, Gee-Hong
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2013 23(24):6773-6776
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7 . Academic Journal
Discovery of fused bicyclic agonists of the orphan G-protein coupled receptor GPR119 with in vivo activity in rodent models of glucose control
저자
by
Semple, Graeme
;
Ren, Albert
;
Fioravanti, Beatriz
;
Pereira, Guillherme
;
Calderon, Imelda
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(10):3134-3141
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7 . Academic Journal
Synthesis and discovery of 2,3-dihydro-3,8-diphenylbenzo[1,4]oxazines as a novel class of potent cholesteryl ester transfer protein inhibitors
저자
by
Wang, Aihua
;
Prouty, Catherine P.
;
Pelton, Patricia D.
;
Yong, Maria
;
Demarest, Keith T.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(4):1432-1435
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7 . Academic Journal
Design and synthesis of potent inhibitors of cholesteryl ester transfer protein (CETP) exploiting a 1,2,3,4-tetrahydroquinoline platform
저자
by
Rano, Thomas A.
;
Sieber-McMaster, Ellen
;
Pelton, Patricia D.
;
Yang, Maria
;
Demarest, Keith T.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(9):2456-2460
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7 . Academic Journal
Design and synthesis of indane-ureido-thioisobutyric acids: A novel class of PPARα agonists
저자
by
Matthews, Jay M.
;
Chen, Xiaoli
;
Cryan, Ellen
;
Hlasta, Dennis J.
;
Rybczynski, Philip J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(24):6773-6778
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