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1 . Academic Journal
Design, synthesis and biological evaluation of Thiazolo[3, 2-a]Pyrimidine derivatives as novel RNase H inhibitors
저자
by
Zhao, Ke-Xin
;
Zhang, Yi-Ying
;
Wang, Jin-Si
;
Wang, Shuai
;
Corona, Angela
, et al.
소스
In
Bioorganic Chemistry
July 2024 148
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7 . Academic Journal
Design and optimization of piperidine-substituted thiophene[3,2-d]pyrimidine-based HIV-1 NNRTIs with improved drug resistance and pharmacokinetic profiles
저자
by
Sun, Yanying
;
Zhou, Zhenzhen
;
Shi, Zhongling
;
Zhao, Fabao
;
Xie, Minghui
, et al.
소스
In
Acta Pharmaceutica Sinica B
July 2024 14(7):3110-3124
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7 . Academic Journal
Discovery of potent HIV-1 NNRTIs by CuAAC click-chemistry-based miniaturized synthesis, rapid screening and structure optimization
저자
by
Jing, Lanlan
;
Wu, Gaochan
;
Zhao, Fabao
;
Jiang, Xiangyi
;
Liu, Na
, et al.
소스
In
European Journal of Medicinal Chemistry
5 November 2024 277
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7 . Academic Journal
Structure-based discovery of novel piperidine-biphenyl-DAPY derivatives as non-nucleoside reverse transcriptase inhibitors featuring improved potency, safety, and selectivity: From piperazine-biphenyl-DAPYs to piperidine-biphenyl-DAPYs
저자
by
Huang, Wen-Juan
;
Pannecouque, Christophe
;
De Clercq, Erik
;
Wang, Shuai
;
Chen, Fen-Er
.
소스
In
European Journal of Medicinal Chemistry
5 October 2024 276
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7 . Academic Journal
Unachieved antiviral strategies with acyclic nucleoside phosphonates: Dedicated to the memory of dr. Salvatore “Sam” Joseph Enna
저자
by
De Clercq, Erik
;
Li, Guangdi
;
Zhang, Yun
;
Huang, Jie
;
Tan, Li
.
소스
In
Biochemical Pharmacology
October 2024 228
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7 . Academic Journal
A scientific career from the early 1960s till 2023: A tale of the various protagonists
저자
by
De Clercq, Erik
.
소스
In
Biochemical Pharmacology
October 2024 228
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3 . Academic Journal
Structure-guided design of novel biphenyl-quinazoline derivatives as potent non-nucleoside reverse transcriptase inhibitors featuring improved anti-resistance, selectivity, and solubility
저자
by
Wang, Jin-Si
;
Zhao, Ke-Xin
;
Zhang, Kun
;
Pannecouque, Christophe
;
De Clercq, Erik
, et al.
소스
In
Bioorganic Chemistry
June 2024 147
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7 . Academic Journal
Design, synthesis, and biological evaluation of benzo[4,5]thieno[2,3-d]pyrimidine derivatives as novel HIV-1 NNRTIs
저자
by
Meng, Bairu
;
Zhuo, Zongji
;
Yu, Han
;
Tao, Sining
;
Chen, Zixuan
, et al.
소스
In
Chinese Chemical Letters
June 2024 35(6)
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7 . Academic Journal
Structure-based design and optimization lead to the identification of novel dihydrothiopyrano[3,2-d]pyrimidine derivatives as potent HIV-1 inhibitors against drug-resistant variants
저자
by
Wang, Zhao
;
Zhang, Heng
;
Gao, Zhen
;
Sang, Zihao
;
De Clercq, Erik
, et al.
소스
In
Acta Pharmaceutica Sinica B
March 2024 14(3):1257-1282
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7 . Academic Journal
In situ click chemistry-based discovery of 1,2,3-triazole-derived diarylpyrimidines as novel HIV-1 NNRTIs by exploiting the tolerant region I in binding pocket
저자
by
Sun, Yanying
;
Feng, Da
;
Zhou, Zhenzhen
;
Zhang, Tao
;
De Clercq, Erik
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 December 2023 96
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