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1 .
Route Optimization of the Non-covalent Modulator of Hemoglobin PF-07059013 for the Treatment of Sickle Cell Disease, Part I: From Discovery Synthesis to First Kilogram-Scale Manufacture
저자
by
Aaron Baldwin
;
Shawn Cabral
;
Kris N. Jones
;
Jeffrey T. Kohrt
;
Chris Limberakis
, et al.
소스
Organic Process Research & Development
. 27:854-865
Web of Science
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7 .
A Small-Molecule Oral Agonist of the Human Glucagon-like Peptide-1 Receptor
저자
by
David A. Griffith
;
David J. Edmonds
;
Jean-Philippe Fortin
;
Amit S. Kalgutkar
;
J. Brent Kuzmiski
, et al.
소스
Journal of medicinal chemistry
. 65(12)
Open Access (OpenAIRE)
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7 .
PF-07059013: A Noncovalent Modulator of Hemoglobin for Treatment of Sickle Cell Disease
저자
by
Ariamala Gopalsamy
;
Ann E. Aulabaugh
;
Amey Barakat
;
Kevin C. Beaumont
;
Shawn Cabral
, et al.
소스
Journal of Medicinal Chemistry
. 64:326-342
Open Access (OpenAIRE)
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7 .
Recent Advances in Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) Inhibitors
저자
by
Chris Limberakis
;
David W. Piotrowski
.
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4 .
RASS‐Enabled S/P−C and S−N Bond Formation for DEL Synthesis
저자
by
Dillon T. Flood
;
Xuejing Zhang
;
Xiang Fu
;
Zhenxiang Zhao
;
Shota Asai
, et al.
소스
Angewandte Chemie
. 132:7447-7453
Full Text (Wiley)
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7 .
Merging C(sp3)–H activation with DNA-encoding
저자
by
David W. Piotrowski
;
Jason S. Chen
;
Mark Edward Flanagan
;
Zhe Zhuang
;
Peng-Xiang Shen
, et al.
소스
Chemical Science
. 11:12282-12288
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7 .
N → N’ acyl migration in the context of a medicinal chemistry program
저자
by
Dennis Anderson
;
Guoyun Bai
;
Shawn Cabral
;
David W. Piotrowski
;
Liuqing Wei
.
소스
Tetrahedron
. 123:132950
Web of Science
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7 .
Acylative Dynamic Kinetic Resolution of Secondary Alcohols: Tandem Catalysis by HyperBTM and Bäckvall's Ruthenium Complex
저자
by
Ahmad Omar Khaled
;
David W. Piotrowski
;
Simonas Balkaitis
;
Edgars Suna
;
Artis Kinens
.
소스
The Journal of organic chemistry
. 86(10)
Scopus
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7 .
PF-07059013: A non-covalent hemoglobin modulator favorably impacts disease state in a mouse model of sickle cell disease
저자
by
Jay M. Janz
;
David W. Piotrowski
;
Dharani Rao
;
Christine Bulawa
;
Zane Wenzel
, et al.
소스
American Journal of Hematology
Full Text (Wiley)
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7 .
Overcoming the Challenges of Making a Single Enantiomer N-1 Substituted Tetrazole Prodrug Using a Tin-Mediated Alkylation and Enzymatic Resolution
저자
by
Anne Akin
;
Asaad S. Nematalla
;
Kevin E. Henegar
;
Javier Magano
;
Thomas A. Brandt
, et al.
소스
Organic Process Research & Development
. 23:1167-1177
Web of Science
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