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1 .
Discovery and Optimization of Potent, Selective, and Brain-Penetrant 1-Heteroaryl-1H-Indazole LRRK2 Kinase Inhibitors for the Treatment of Parkinson’s Disease
저자
by
David A. Candito
;
Vladimir Simov
;
Anmol Gulati
;
Solomon Kattar
;
Ryan W. Chau
, et al.
소스
Journal of Medicinal Chemistry
. 65:16801-16817
Web of Science
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7 .
Racemic Synthesis of a Key 1,4-Dihydro-2H-spiro[isoquinoline-3,4′-piperidin]-3′-ol Building Block
저자
by
David A. Candito
;
Theodore A. Martinot
;
Jing Su
;
Josep Saurí
;
Yu-hong Lam
, et al.
소스
Organic Process Research & Development
. 26:3034-3041
Web of Science
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7 .
Synthetic Studies Probing Elansolid Biosynthesis: A para -Quinone-Methide-Triggered Intramolecular Diels-Alder Reaction
저자
by
Liang-Liang Wang
;
Andreas Kirschning
;
Gerald Dräger
;
David A. Candito
.
소스
European Journal of Organic Chemistry
. 2017:5582-5591
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6 . Academic Journal
Formal Synthesis of Nitidine and NK109 via Palladium-Catalyzed Domino Direct Arylation/N-Arylation of Aryl Triflates.
저자
by
Mathieu Blanchot
;
David A. Candito
;
Florent Larnaud
;
Mark Lautens
.
소스
Organic Letters
. Mar2011, Vol. 13 Issue 6, p1486-1489. 4p.
Full Text (ACS)
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6 . Academic Journal
Exploiting the Chemistry of Strained Rings: Synthesis of Indoles via Domino Reaction of Aryl Iodides with 2H-Azirines.
저자
by
David A. Candito
;
Mark Lautens
.
소스
Organic Letters
. Aug2010, Vol. 12 Issue 15, p3312-3315. 4p.
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4 .
Harnessing a p-Quinone Methide Intermediate in the Biomimetic Total Synthesis of the Highly Active Antibiotic 20-Deoxy-Elansolid B1
저자
by
Jennifer Herrmann
;
Rolf Müller
;
Andreas Kirschning
;
Gerald Dräger
;
David A. Candito
, et al.
소스
Chemistry (Weinheim an der Bergstrasse, Germany)
. 23(22)
Full Text (Wiley)
Scopus
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7 .
A Bio-Chemosynthetic Approach to Superparamagnetic Iron Oxide-Ansamitocin Conjugates for Use in Magnetic Drug Targeting
저자
by
Andreas Kirschning
;
Nadja-Carola Bigall
;
Jan F. Miethe
;
Yu Xie
;
Asha Balakrishnan
, et al.
소스
Chemistry (Weinheim an der Bergstrasse, Germany)
. 23(10)
Full Text (Wiley)
Scopus
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7 . Academic Journal
Palladium-Catalyzed Reductive ortho-Arylation: Evidence for the Decomposition of 1,2-Dimethoxyethane and Subsequent Arylpalladium(II) Reduction.
저자
by
Andrew Martins
;
David A. Candito
;
Mark Lautens
.
소스
Organic Letters
. Nov2010, Vol. 12 Issue 22, p5186-5188. 3p.
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5 .
Intramolecular Aryne–Ene Reaction: Synthetic and Mechanistic Studies
저자
by
Jane Panteleev
;
David A. Candito
;
Mark Lautens
.
소스
Journal of the American Chemical Society
. 133:14200-14203
Web of Science
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5 .
Formal Synthesis of Nitidine and NK109 via Palladium-Catalyzed Domino Direct Arylation/N-Arylation of Aryl Triflates
저자
by
Florent Larnaud
;
David A. Candito
;
Mathieu Blanchot
;
Mark Lautens
.
소스
Organic Letters
. 13:1486-1489
Web of Science
Scopus
JCR 저널정보
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