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1 . Academic Journal
Screening a protein kinase inhibitor library against Plasmodium falciparum
저자
by
Irene Hallyburton
;
Raffaella Grimaldi
;
Andrew Woodland
;
Beatriz Baragaña
;
Torsten Luksch
, et al.
소스
Malaria Journal, Vol 16, Iss 1, Pp 1-11 (2017)
Open Access (DOAJ)
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7 .
Identification and Optimization of a Series of 8-Hydroxy Naphthyridines with Potent In Vitro Antileishmanial Activity: Initial SAR and Assessment of In Vivo Activity
저자
by
Michael G. Thomas
;
Maria L. Marco
;
John Thomas
;
Daniel Spinks
;
Ian H. Gilbert
, et al.
소스
Journal of Medicinal Chemistry
. 63:9523-9539
Open Access (OpenAIRE)
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7 .
2,4-Diamino-6-methylpyrimidines for the potential treatment of Chagas’ disease
저자
by
Manu De Rycker
;
John Thomas
;
Michael G. Thomas
;
Timothy J. Miles
;
Paul G. Wyatt
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 28:3025-3030
Open Access (OpenAIRE)
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7 .
Discovery and Optimization of 5-Amino-1,2,3-triazole-4-carboxamide Series against Trypanosoma cruzi
저자
by
Laste Stojanovski
;
Tania Bakshi
;
Iain H. Reid
;
Maria L. Marco
;
Stephen Brand
, et al.
소스
Journal of Medicinal Chemistry
Open Access (OpenAIRE)
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7 . Academic Journal
One Scaffold, Three Binding Modes: Novel and Selective Pteridine Reductase 1 Inhibitors Derived from Fragment Hits Discovered by Virtual Screening.
저자
by
Chidochangu P. Mpamhanga
;
Daniel Spinks
;
Lindsay B. Tulloch
;
Emma J. Shanks
;
David A. Robinson
, et al.
소스
Journal of Medicinal Chemistry
. Jul2009, Vol. 52 Issue 14, p4454-4465. 12p.
Full Text (ACS)
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7 .
Discovery of a Novel Class of Orally Active Trypanocidal N-Myristoyltransferase Inhibitors
저자
by
David A. Robinson
;
Suzanne Norval
;
Irene Hallyburton
;
Stephen Brand
;
Ian H. Gilbert
, et al.
소스
Journal of Medicinal Chemistry
Open Access (OpenAIRE)
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7 .
Optimisation of the Anti-Trypanosoma brucei Activity of the Opioid Agonist U50488
저자
by
Alan H. Fairlamb
;
Victoria Smith
;
Daniel Spinks
;
Julie A. Frearson
;
Ruth Brenk
, et al.
소스
Chemmedchem
Open Access (OpenAIRE)
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7 .
Design, Synthesis and Biological Evaluation of Novel Inhibitors ofTrypanosoma bruceiPteridine Reductase 1
저자
by
David A. Robinson
;
Alan H. Fairlamb
;
Ian H. Gilbert
;
Iain T. Collie
;
Han B. Ong
, et al.
소스
Chemmedchem
Open Access (OpenAIRE)
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7 .
Chemical Validation of Trypanothione Synthetase
저자
by
Paul G. Wyatt
;
Alan H. Fairlamb
;
Julie A. Frearson
;
Sandra L. Oza
;
Stephen Thompson
, et al.
소스
Journal of Biological Chemistry
. 284:36137-36145
Full Text (ScienceDirect O/A)
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7 .
One Scaffold, Three Binding Modes: Novel and Selective Pteridine Reductase 1 Inhibitors Derived from Fragment Hits Discovered by Virtual Screening†
저자
by
David A. Robinson
;
William N. Hunter
;
Emma Shanks
;
Alan H. Fairlamb
;
Ian H. Gilbert
, et al.
소스
Journal of Medicinal Chemistry
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