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1 .
Discovery of the Migraine Prevention Therapeutic Aimovig (Erenumab), the First FDA-Approved Antibody against a G-Protein-Coupled Receptor
저자
by
Brian Mingtung Chan
;
Kelly A Berry
;
David W. Brankow
;
Chadwick T. King
;
Sylvia Nai-Yu Hu
, et al.
소스
ACS Pharmacol Transl Sci
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7 . Academic Journal
Identification of Potent, Selective, and Metabolically Stable Peptide Antagonists to the Calcitonin Gene-Related Peptide (CGRP) Receptor.
저자
by
Les P. Miranda
;
Jerry Ryan Holder
;
Licheng Shi
;
Brian Bennett
;
Jennifer Aral
, et al.
소스
Journal of Medicinal Chemistry
. Dec2008, Vol. 51 Issue 24, p7889-7897. 9p.
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7 . Academic Journal
Design and Synthesis of Conformationally Constrained Glucagon-Like Peptide-1 Derivatives with Increased Plasma Stability and Prolonged in Vivo Activity.
저자
by
Les P. Miranda
;
Katherine A. Winters
;
Colin V. Gegg
;
Ankita Patel
;
Jennifer Aral
, et al.
소스
Journal of Medicinal Chemistry
. Apr2008, Vol. 51 Issue 9, p2758-2765. 8p.
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7 .
Pharmaceutical Optimization of Peptide Toxins for Ion Channel Targets: Potent, Selective, and Long-Lived Antagonists of Kv1.3
저자
by
Kevin Gaida
;
Xuxia Zhang
;
Robin Elliott
;
Benxian Liu
;
Andrea Itano
, et al.
소스
Journal of Medicinal Chemistry
. 58:6784-6802
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7 .
Peptide antagonists of the calcitonin gene-related peptide (CGRP) receptor with improved pharmacokinetics and pharmacodynamics
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by
Eileen Johnson
;
Jerry Ryan Holder
;
Barton H. Manning
;
Licheng Shi
;
Kevin Salyers
, et al.
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Biopolymers
. 100:422-430
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7 .
Ligand-Binding Mass Spectrometry to Study Biotransformation of Fusion Protein Drugs and Guide Immunoassay Development: Strategic Approach and Application to Peptibodies Targeting the Thrombopoietin Receptor
저자
by
Michael Hall
;
Hsieng Sen Lu
;
Christopher S. Spahr
;
Robert Ortiz
;
Steven Yu
, et al.
소스
The AAPS Journal
. 12:576-585
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7 .
Investigation of the effects of altered receptor binding activity on the clearance of erythropoiesis-stimulating proteins: Nonerythropoietin receptor-mediated pathways may play a major role
저자
by
Linda O. Narhi
;
Graham Molineux
;
Sameer Doshi
;
Balaji Agoram
;
Ken Aoki
, et al.
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Journal of Pharmaceutical Sciences
. 98:2198-2211
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7 .
Interactions between PEG and type I soluble tumor necrosis factor receptor: Modulation by pH and by PEGylation at the N terminus
저자
by
Giovanni B. Strambini
;
Margherita Gonnelli
;
Byeong S. Chang
;
Bruce A. Kerwin
;
Colin V. Gegg
, et al.
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Protein Science
. 11:1825-1833
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7 .
An Acyl-Ghrelin-Specific Neutralizing Antibody Inhibits the Acute Ghrelin-Mediated Orexigenic Effects in Mice
저자
by
David W. Brankow
;
Shu-Chen Lu
;
Jing Xu
;
Shuying Liu
;
Shirley Steavenson
, et al.
소스
Molecular Pharmacology
. 75:901-907
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7 .
Identification of Potent, Selective, and Metabolically Stable Peptide Antagonists to the Calcitonin Gene-Related Peptide (CGRP) Receptor
저자
by
Licheng Shi
;
Jennifer Aral
;
Richard S. Rogers
;
Violeta G. Valladares
;
Hongyan Li
, et al.
소스
Journal of Medicinal Chemistry
. 51:7889-7897
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