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1 .
Discovery of (2R)-N-[3-[2-[(3-Methoxy-1-methyl-pyrazol-4-yl)amino]pyrimidin-4-yl]-1H-indol-7-yl]-2-(4-methylpiperazin-1-yl)propenamide (AZD4205) as a Potent and Selective Janus Kinase 1 Inhibitor
저자
by
Nanhua Deng
;
Sameer Kawatkar
;
Haoyu Wang
;
Michael Zinda
;
Allan Wu
, et al.
소스
Journal of Medicinal Chemistry
. 63:4517-4527
Web of Science
Scopus
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7 .
Discovery of CC-99677, a selective targeted covalent MAPKAPK2 (MK2) inhibitor for autoimmune disorders
저자
by
JOHN Malona
;
CLAUDIO CHUAQUI
;
BORIS M. SELETSKY
;
LISA BEEBE
;
SUSAN CANTIN
, et al.
소스
Translational research : the journal of laboratory and clinical medicine
. 249
Open Access (OpenAIRE)
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7 .
Discovery of SY-5609: A Selective, Noncovalent Inhibitor of CDK7
저자
by
Ashraf Wilsily
;
Robert Zahler
;
Nan Ke
;
Claudio Chuaqui
;
Michael J. Bradley
, et al.
소스
Journal of medicinal chemistry
. 65(2)
Open Access (OpenAIRE)
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7 .
Abstract 5393: An oral and selective CDK12 inhibitor demonstrates robust anti-tumor activity
저자
by
Shan hu
;
David Moebius
;
Wojciech Dworakowski
;
Elliott Cooper
;
Derek LaPlaca
, et al.
소스
Cancer Research
. 82:5393-5393
Full Text (AACR)
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7 .
Discovery and Optimization of a Novel Series of Highly Selective JAK1 Kinase Inhibitors
저자
by
Haixia Wang
;
Marat Alimzhanov
;
Paul Lyne
;
Jason Grant Kettle
;
Jie Shi
, et al.
소스
Journal of Medicinal Chemistry
. 61:5235-5244
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7 .
Utilization of Structure-Based Design to Identify Novel, Irreversible Inhibitors of EGFR Harboring the T790M Mutation
저자
by
Darren Cross
;
Lakshmaiah Gingipalli
;
Teresa Klinowska
;
Cath Eberlein
;
Nicola Colclough
, et al.
소스
ACS Medicinal Chemistry Letters
. 7:514-519
Open Access (OpenAIRE)
Web of Science
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7 .
Potent and Selective CK2 Kinase Inhibitors with Effects on Wnt Pathway Signaling in Vivo
저자
by
Emma Jenkins
;
Larry Bao
;
Christopher R. Denz
;
Andrew D. Ferguson
;
Geoff Holdgate
, et al.
소스
ACS Medicinal Chemistry Letters
. 7:300-305
Open Access (OpenAIRE)
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7 .
Identification of azabenzimidazoles as potent JAK1 selective inhibitors
저자
by
Jon Read
;
Haixia Wang
;
Dennis Huszar
;
Sameer Kawatkar
;
Kelly Goodwin
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 26:60-67
Web of Science
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7 .
Correction to Discovery of Pyrazolo[1,5-a]pyrimidine B-Cell Lymphoma 6 (BCL6) Binders and Optimization to High Affinity Macrocyclic Inhibitors
저자
by
William McCoull
;
Roman D. Abrams
;
Erica Anderson
;
Kevin Blades
;
Peter Barton
, et al.
소스
Journal of medicinal chemistry
. 60(14)
Open Access (OpenAIRE)
Scopus
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7 .
Discovery of Pyrazolo[1,5-a]pyrimidine B-Cell Lymphoma 6 (BCL6) Binders and Optimization to High Affinity Macrocyclic Inhibitors
저자
by
Jennifer E. Nelson
;
Graeme R. Robb
;
Martin R. Howard
;
Piotr Raubo
;
Paul D. Kemmitt
, et al.
소스
Journal of medicinal chemistry
. 60(10)
Open Access (OpenAIRE)
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