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1 . Academic Journal
Phase II study investigating the efficacy and safety of glesatinib (MGCD265) in patients with advanced NSCLC containing MET activating alterations
저자
by
Hong, David S.
;
Cappuzzo, Federico
;
Chul Cho, Byoung
;
Dowlati, Afshin
;
Hussein, Maen
, et al.
소스
In
Lung Cancer
April 2024 190
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7 . Academic Journal
Adeno-to-squamous transition drives resistance to KRAS inhibition in LKB1 mutant lung cancer
저자
by
Tong, Xinyuan
;
Patel, Ayushi S.
;
Kim, Eejung
;
Li, Hongjun
;
Chen, Yueqing
, et al.
소스
In
Cancer Cell
11 March 2024 42(3):413-428
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7 . Academic Journal
Design and evaluation of achiral, non-atropisomeric 4-(aminomethyl)phthalazin-1(2H)-one derivatives as novel PRMT5/MTA inhibitors
저자
by
Smith, Christopher R.
;
Aranda, Ruth
;
Christensen, James G.
;
Engstrom, Lars D.
;
Gunn, Robin J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 October 2022 71
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7 . Academic Journal
Discovery of Five SOS2 Fragment Hits with Binding Modes Determined by SOS2 X‑Ray Cocrystallography.
저자
by
Smith, Christopher R.
;
Chen, Dan
;
Christensen, James G.
;
Coulombe, René
;
Féthière, James
, et al.
소스
Journal of Medicinal Chemistry; 1/11/2024, Vol. 67 Issue 1, p774-781, 8p
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7 . Academic Journal
Intracranial Efficacy of Adagrasib in Patients From the KRYSTAL-1 Trial With KRAS G12C -Mutated Non–Small-Cell Lung Cancer Who Have Untreated CNS Metastases.
저자
by
Negrao, Marcelo V.
;
Spira, Alexander I.
;
Heist, Rebecca S.
;
Jänne, Pasi A.
;
Pacheco, Jose M.
, et al.
소스
Journal of Clinical Oncology; 10/1/2023, Vol. 41 Issue 28, p4472-4477, 8p
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7 . Academic Journal
HGF/c-Met pathway is one of the mediators of sunitinib-induced tumor cell type-dependent metastasis
저자
by
Shojaei, Farbod
;
Simmons, Brett H.
;
Lee, Joseph H.
;
Lappin, Patrick B.
;
Christensen, James G.
.
소스
In
Cancer Letters
1 July 2012 320(1):48-55
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7 . Academic Journal
Preexistence and Clonal Selection of MET Amplification in EGFR Mutant NSCLC
저자
by
Turke, Alexa B.
;
Zejnullahu, Kreshnik
;
Wu, Yi-Long
;
Song, Youngchul
;
Dias-Santagata, Dora
, et al.
소스
In
Cancer Cell
2010 17(1):77-88
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7 . Academic Journal
Adagrasib with or without Cetuximab in Colorectal Cancer with Mutated KRAS G12C.
저자
by
Yaeger, Rona
;
Weiss, Jared
;
Pelster, Meredith S.
;
Spira, Alexander I.
;
Barve, Minal
, et al.
소스
New England Journal of Medicine
. 1/5/2023, Vol. 388 Issue 1, p44-54. 11p.
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7 . Academic Journal
Phase I Study Evaluating Glesatinib (MGCD265), An Inhibitor of MET and AXL, in Patients with Non-small Cell Lung Cancer and Other Advanced Solid Tumors.
저자
by
Kollmannsberger, Christian
;
Hurwitz, Herbert
;
Bazhenova, Lyudmila
;
Cho, Byoung Chul
;
Hong, David
, et al.
소스
Targeted Oncology; Jan2023, Vol. 18 Issue 1, p105-118, 14p
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7 . Academic Journal
c-Met as a target for human cancer and characterization of inhibitors for therapeutic intervention
저자
by
Christensen, James G.
;
Burrows, Jon
;
Salgia, Ravi
.
소스
In
Cancer Letters
2005 225(1):1-26
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