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1 . Academic Journal
Pharmacophore hybridization approach to discover novel pyrazoline-based hydantoin analogs with anti-tumor efficacy
저자
by
Upadhyay, Neha
;
Tilekar, Kalpana
;
Loiodice, Fulvio
;
Anisimova, Natalia Yu.
;
Spirina, Tatiana S.
, et al.
소스
In
Bioorganic Chemistry
February 2021 107
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7 . Academic Journal
Power of two: combination of therapeutic approaches involving glucose transporter (GLUT) inhibitors to combat cancer
저자
by
Tilekar, Kalpana
;
Upadhyay, Neha
;
Iancu, Cristina V.
;
Pokrovsky, Vadim
;
Choe, Jun-yong
, et al.
소스
In
BBA - Reviews on Cancer
December 2020 1874(2)
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7 . Academic Journal
Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential
저자
by
Tilekar, Kalpana
;
Upadhyay, Neha
;
Hess, Jessica D.
;
Macias, Lucasantiago Henze
;
Mrowka, Piotr
, et al.
소스
In
European Journal of Medicinal Chemistry
15 September 2020 202
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7 . Academic Journal
Electrochemical and Structural Study of the Buried Tryptophan in Azurin: Effects of Hydration and Polarity on the Redox Potential of W48.
저자
by
Tyson, Kristin
;
Tangtartharakul, Chanin B.
;
Zeug, Matthias
;
Findling, Nathan
;
Haddy, Alice
, et al.
소스
Journal of Physical Chemistry B; 12/21/202, Vol. 127 Issue 50, p133-143, 11p
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7 . Academic Journal
Discrimination of GLUTs by Fructose Isomers Enables Simultaneous Screening of GLUT5 and GLUT2 Activity in Live Cells.
저자
by
Gora, Nazar
;
Weselinski, Lukasz J.
;
Begoyan, Vagarshak V.
;
Cooper, Andrew
;
Choe, Jun-yong
, et al.
소스
ACS Chemical Biology; 5/19/2023, Vol. 18 Issue 5, p1089-1100, 12p
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7 . Academic Journal
GLUT3 inhibitor discovery through in silico ligand screening and in vivo validation in eukaryotic expression systems.
저자
by
Iancu, Cristina V.
;
Bocci, Giovanni
;
Ishtikhar, Mohd
;
Khamrai, Moumita
;
Oreb, Mislav
, et al.
소스
Scientific Reports
. 1/26/2022, Vol. 12 Issue 1, p1-13. 13p.
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7 . Academic Journal
Identification of new GLUT2-selective inhibitors through in silico ligand screening and validation in eukaryotic expression systems.
저자
by
Schmidl, Sina
;
Ursu, Oleg
;
Iancu, Cristina V.
;
Oreb, Mislav
;
Oprea, Tudor I.
, et al.
소스
Scientific Reports
. 7/2/2021, Vol. 11 Issue 1, p1-12. 12p.
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7 . Academic Journal
Crystal structures of non-oxidative decarboxylases reveal a new mechanism of action with a catalytic dyad and structural twists.
저자
by
Zeug, Matthias
;
Markovic, Nebojsa
;
Iancu, Cristina V.
;
Tripp, Joanna
;
Oreb, Mislav
, et al.
소스
Scientific Reports
. 2/4/2021, Vol. 11 Issue 1, p1-13. 13p.
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7 . Academic Journal
A label-free real-time method for measuring glucose uptake kinetics in yeast.
저자
by
Schmidl, Sina
;
Iancu, Cristina V
;
Reifenrath, Mara
;
Choe, Jun-yong
;
Oreb, Mislav
.
소스
FEMS Yeast Research
. Feb2021, Vol. 21 Issue 1, p1-8. 8p.
Open Access (OUP)
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7 . Academic Journal
Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine‐2,5‐dione Hybrids as Potential Antitumor Agents.
저자
by
Tilekar, Kalpana
;
Upadhyay, Neha
;
Meyer‐Almes, Franz‐Josef
;
Loiodice, Fulvio
;
Anisimova, Natalia Y.
, et al.
소스
ChemMedChem; 10/5/2020, Vol. 15 Issue 19, p1813-1825, 13p
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