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1 . Academic Journal
Polo-like Kinase 2 (PLK2) Phosphorylates α-Synuclein at Serine 129 in Central Nervous System
저자
by
Inglis, Kelly J.
;
Chereau, David
;
Brigham, Elizabeth F.
;
Chiou, San-San
;
Schöbel, Susanne
, et al.
소스
In
Journal of Biological Chemistry
30 January 2009 284(5):2598-2602
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7 . Academic Journal
Discovery of 4-alkylamino-7-aryl-3-cyanoquinoline LRRK2 kinase inhibitors
저자
by
Garofalo, Albert W.
;
Adler, Marc
;
Aubele, Danielle L.
;
Brigham, Elizabeth F.
;
Chian, David
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 April 2013 23(7):1974-1977
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7 . Academic Journal
Novel Piperidinyl-Azetidines as Potent and Selective CCR4 Antagonists Elicit Antitumor Response as a Single Agent and in Combination with Checkpoint Inhibitors.
저자
by
Robles, Omar
;
Jackson, Jeffrey J.
;
Marshall, Lisa
;
Talay, Oezcan
;
Chian, David
, et al.
소스
Journal of Medicinal Chemistry; 8/13/2020, Vol. 63 Issue 15, p8584-8607, 24p
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7 . Academic Journal
Discovery of a Potent and Selective CCR4 Antagonist That Inhibits T
reg
Trafficking into the Tumor Microenvironment.
저자
by
Jackson, Jeffrey J.
;
Ketcham, John M.
;
Younai, Ashkaan
;
Abraham, Betty
;
Biannic, Berenger
, et al.
소스
Journal of Medicinal Chemistry; 7/11/2019, Vol. 62 Issue 13, p6190-6213, 24p
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7 . Academic Journal
Design of an orally efficacious hydroxyethylamine (HEA) BACE-1 inhibitor in a preclinical animal model
저자
by
Truong, Anh P.
;
Tóth, Gergley
;
Probst, Gary D.
;
Sealy, Jennifer M.
;
Bowers, Simeon
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(21):6231-6236
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7 . Periodical
Discovery of a Potent and Selective CCR4 Antagonist That Inhibits TregTrafficking into the Tumor Microenvironment
저자
by
Jackson, Jeffrey J.
;
Ketcham, John M.
;
Younai, Ashkaan
;
Abraham, Betty
;
Biannic, Berenger
, et al.
소스
Journal of Medicinal Chemistry; July 2019, Vol. 62 Issue: 13 p6190-6213, 24p
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7 . Academic Journal
Variable effects of the gamma-secretase inhibitor ELND006 on Aβ across different compartments (brain, ISF, CSF, and plasma) following sustained exposure via subcutaneous osmotic pumps in wild-type mice
저자
by
Brigham, Elizabeth
;
Wong, Angelina
;
Rampurna, Gullapalli
;
Quinn, Kevin
;
Kwong, Grace
, et al.
소스
In
Alzheimer's & Dementia: The Journal of the Alzheimer's Association
July 2011 7(4) Supplement:S313-S314
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7 . Academic Journal
Tumors establish resistance to immunotherapy by regulating T-reg recruitment via CCR4
저자
by
Marshall, Lisa A.
;
Marubayashi, Sachie
;
Jorapur, Aparna
;
Jacobson, Scott
;
Zibinsky, Mikhail
, et al.
소스
JOURNAL FOR IMMUNOTHERAPY OF CANCER
; 2020, 8 2, pe000764 11p.
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7 . Academic Journal
Discovery and optimization of potent and selective inhibitors of USP7 to enhance anti-tumor immunity and target tumor growth
저자
by
Abraham, Betty
;
Adusumilli, Lavanya
;
Biannic, Berenger
;
Bradford, Delia
;
Brovarney, Martin
, et al.
소스
CANCER RESEARCH
; JUL 2018, 78 13, 3p. Supplement: S
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7 . Academic Journal
Potent and selective next generation inhibitors of indoleamine-2,3-dioxygenase (IDO1) for the treatment of cancer
저자
by
Powers, Jay P.
;
Walters, Matthew J.
;
Noubade, Rajkumar
;
Young, Stephen W.
;
Marshall, Lisa
, et al.
소스
CANCER RESEARCH
; AUG 1 2015, 75 3p. Supplement: 15
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