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1 . Academic Journal
5-HT6 receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivatives
저자
by
Drop, Marcin
;
Koczurkiewicz-Adamczyk, Paulina
;
Bento, Ophélie
;
Pietruś, Wojciech
;
Satała, Grzegorz
, et al.
소스
In
European Journal of Medicinal Chemistry
5 September 2024 275
Full Text (ScienceDirect)
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7 . Academic Journal
Neuropathic pain-alleviating activity of novel 5-HT6 receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamide
저자
by
Drop, Marcin
;
Jacquot, Florian
;
Canale, Vittorio
;
Chaumont-Dubel, Severine
;
Walczak, Maria
, et al.
소스
In
Bioorganic Chemistry
October 2021 115
Full Text (ScienceDirect)
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7 . Academic Journal
A dual-acting 5-HT6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties
저자
by
Canale, Vittorio
;
Grychowska, Katarzyna
;
Kurczab, Rafał
;
Ryng, Mateusz
;
Keeri, Abdul Raheem
, et al.
소스
In
European Journal of Medicinal Chemistry
15 December 2020 208
Full Text (ScienceDirect)
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7 . Academic Journal
Novel non-sulfonamide 5-HT6 receptor partial inverse agonist in a group of imidazo[4,5-b]pyridines with cognition enhancing properties
저자
by
Vanda, David
;
Soural, Miroslav
;
Canale, Vittorio
;
Chaumont-Dubel, Séverine
;
Satała, Grzegorz
, et al.
소스
In
European Journal of Medicinal Chemistry
20 January 2018 144:716-729
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7 . Academic Journal
Angiogenin induces modifications in the astrocyte secretome: Relevance to amyotrophic lateral sclerosis
저자
by
Skorupa, Alexandra
;
Urbach, Serge
;
Vigy, Oana
;
King, Matthew A.
;
Chaumont-Dubel, Séverine
, et al.
소스
In
Journal of Proteomics
8 October 2013 91:274-285
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7 . Periodical
Superiority of the Triple-Acting 5-HT6R/5-HT3R Antagonist and MAO-B Reversible Inhibitor PZ-1922over 5-HT6R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Rats
저자
by
Grychowska, Katarzyna
;
López-Sánchez, Uriel
;
Vitalis, Mathieu
;
Canet, Geoffrey
;
Satała, Grzegorz
, et al.
소스
Journal of Medicinal Chemistry; November 2023, Vol. 66 Issue: 21 p14928-14947, 20p
Full Text (ACS)
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7 . Academic Journal
Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT 6 and D 3 R Affinity in the 1 H -Pyrrolo[3,2- c ]quinoline Series.
저자
by
Grychowska, Katarzyna
;
Pietruś, Wojciech
;
Kulawik, Ludmiła
;
Bento, Ophélie
;
Satała, Grzegorz
, et al.
소스
Molecules
. Feb2023, Vol. 28 Issue 3, p1096. 16p.
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7 . Academic Journal
Impact of 5-HT 6 Receptor Subcellular Localization on Its Signaling and Its Pathophysiological Roles.
저자
by
Chaumont-Dubel, Séverine
;
Galant, Sonya
;
Prieur, Matthieu
;
Bouschet, Tristan
;
Bockaert, Joël
, et al.
소스
Cells (2073-4409)
. Feb2023, Vol. 12 Issue 3, p426. 12p.
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7 . Academic Journal
1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT 6 R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity.
저자
by
Canale, Vittorio
;
Trybała, Wojciech
;
Chaumont-Dubel, Séverine
;
Koczurkiewicz-Adamczyk, Paulina
;
Satała, Grzegorz
, et al.
소스
Biomolecules (2218-273X)
. Jan2023, Vol. 13 Issue 1, p12. 16p.
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7 . Academic Journal
Imidazopyridine-Based 5‑HT
6
Receptor Neutral Antagonists: Impact of N
1
‑Benzyl and N
1
‑Phenylsulfonyl Fragments on Different Receptor Conformational States.
저자
by
Vanda, David
;
Canale, Vittorio
;
Chaumont-Dubel, Severine
;
Kurczab, Rafał
;
Satała, Grzegorz
, et al.
소스
Journal of Medicinal Chemistry; 1/28/2021, Vol. 64 Issue 2, p1180-1196, 17p
Full Text (ACS)
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