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1 . Academic Journal
Evaluation of a Competitive Equilibrium Dialysis Approach for Assessing the Impact of Protein Binding on Clearance Predictions
저자
by
Jones, Robert S.
;
Chang, Jae H.
;
Flores, Mauricio
;
Brecht, Elliot
.
소스
In
Journal of Pharmaceutical Sciences
January 2021 110(1):536-542
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6 . Report
Multilevel Second-Moment Methods with Group Decomposition for Multigroup Transport Problems
저자
by
Anistratov, Dmitriy Y.
;
Coale, Joseph M.
;
Warsa, James S.
;
Chang, Jae H.
.
소스
Open Access (Arxiv)
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6 . Academic Journal
High resolution time integration for S N radiation transport
저자
by
Thoreson, Greg
;
McClarren, Ryan G.
;
Chang, Jae H.
.
소스
In
Annals of Nuclear Energy
2009 36(3):263-267
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5 . Book
Chapter 20 - Application of genetically modified rodent models in drug discovery and development for translation of clinical ADME properties
저자
by
Jones, Robert S.
;
Ly, Justin Q.
;
Chang, Jae H.
.
소스
In
Identification and Quantification of Drugs, Metabolites, Drug Metabolizing Enzymes, and Transporters
Edition: Second Edition. 2020:555-594
Full Text (ScienceDirect)
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5 . Academic Journal
Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927
저자
by
Labadie, Sharada S.
;
Li, Jun
;
Blake, Robert A.
;
Chang, Jae H.
;
Goodacre, Simon
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 August 2019 29(16):2090-2093
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7 . Academic Journal
Unexpected equivalent potency of a constrained chromene enantiomeric pair rationalized by co-crystal structures in complex with estrogen receptor alpha
저자
by
Zhang, Birong
;
Kiefer, James R.
;
Blake, Robert A.
;
Chang, Jae H.
;
Hartman, Steven
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 April 2019 29(7):905-911
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7 . Periodical
Analysis of the Bile Acid Composition in a Fibroblast Growth Factor 19-Expressing Liver-Humanized Mouse Model and Its Use for CYP3A4-Mediated Drug–Drug Interaction Studies
저자
by
Mezler, Mario
;
Jones, Robert S.
;
Sangaraju, Dewakar
;
Goldman, Devorah C.
;
Hoffmann, Matthew
, et al.
소스
Drug Metabolism and Disposition; 2023, Vol. 51 Issue: 10 p1391-1402, 12p
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7 . Academic Journal
Discovery of 3,5-substituted 6-azaindazoles as potent pan-Pim inhibitors
저자
by
Hu, Huiyong
;
Wang, Xiaojing
;
Chan, Grace Ka Yan
;
Chang, Jae H.
;
Do, Steven
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 November 2015 25(22):5258-5264
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7 .
Contributors
저자
by
Al Qaraghuli, Farah
;
Alluri, Ravindra Varma
;
Argon, Sophie M.A.
;
Bajaj, Piyush
;
Bapiro, Tashinga E.
, et al.
소스
In
Identification and Quantification of Drugs, Metabolites, Drug Metabolizing Enzymes, and Transporters
Edition: Second Edition. 2020:xi-xiii
Full Text (ScienceDirect)
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7 . Periodical
Application of Empirical Scalars To Enable Early Prediction of Human Hepatic Clearance Using In Vitro-In Vivo Extrapolation in Drug Discovery: An Evaluation of 173 Drugs
저자
by
Jones, Robert S.
;
Leung, Christian
;
Chang, Jae H.
;
Brown, Suzanne
;
Liu, Ning
, et al.
소스
Drug Metabolism and Disposition; 2022, Vol. 50 Issue: 8 p1053-1063, 11p
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