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1 . Academic Journal
An evolutionarily conserved N-terminal leucine is essential for MX1 GTPase antiviral activity against different families of RNA viruses
저자
by
McKellar, Joe
;
Arnaud-Arnould, Mary
;
Chaloin, Laurent
;
Tauziet, Marine
;
Arpin-André, Charlotte
, et al.
소스
In
Journal of Biological Chemistry
January 2023 299(1)
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7 . Academic Journal
4-Substituted-1,2,3-triazolo nucleotide analogues as CD73 inhibitors, their synthesis, in vitro screening, kinetic and in silico studies
저자
by
Ghoteimi, Rayane
;
Braka, Abdennour
;
Rodriguez, Céline
;
Cros-Perrial, Emeline
;
Tai Nguyen, Van
, et al.
소스
In
Bioorganic Chemistry
February 2021 107
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7 . Academic Journal
Lead optimization and biological evaluation of fragment-based cN-II inhibitors
저자
by
Guillon, Rémi
;
Rahimova, Rahila
;
Preeti
;
Egron, David
;
Rouanet, Sonia
, et al.
소스
In
European Journal of Medicinal Chemistry
15 April 2019 168:28-44
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7 . Academic Journal
The IbeA protein from adherent invasive Escherichia coli is a flavoprotein sharing structural homology with FAD‐dependent oxidoreductases.
저자
by
Paris, Théo
;
Kiss, Agneta
;
Signor, Luca
;
Lutfalla, Georges
;
Blaise, Mickaël
, et al.
소스
FEBS Journal
. Jan2024, Vol. 291 Issue 1, p177-203. 27p.
Full Text (Wiley)
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7 . Academic Journal
Structure–activity relationships of β-hydroxyphosphonate nucleoside analogues as cytosolic 5′-nucleotidase II potential inhibitors: Synthesis, in vitro evaluation and molecular modeling studies
저자
by
Meurillon, Maïa
;
Marton, Zsuzsanna
;
Hospital, Audrey
;
Jordheim, Lars Petter
;
Béjaud, Jérôme
, et al.
소스
In
European Journal of Medicinal Chemistry
22 April 2014 77:18-37
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7 . Academic Journal
Selectivity of kinases on the activation of tenofovir, an anti-HIV agent
저자
by
Varga, Andrea
;
Gráczer, Éva
;
Chaloin, Laurent
;
Liliom, Károly
;
Závodszky, Péter
, et al.
소스
In
European Journal of Pharmaceutical Sciences
23 January 2013 48(1-2):307-315
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7 . Academic Journal
Synthesis of ( R)- and ( S)-β-hydroxyphosphonate acyclonucleosides: structural analogues of Adefovir (PMEA)
저자
by
Kasthuri, Mahesh
;
Chaloin, Laurent
;
Périgaud, Christian
;
Peyrottes, Suzanne
.
소스
In
Tetrahedron: Asymmetry
2011 22(14):1505-1511
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6 . Academic Journal
Second‐Generation CD73 Inhibitors Based on a 4,6‐Biaryl‐2‐thiopyridine Scaffold.
저자
by
Ghoteimi, Rayane
;
Braka, Abdennour
;
Rodriguez, Céline
;
Cros‐Perrial, Emeline
;
Duvauchelle, Valentin
, et al.
소스
ChemMedChem; 4/3/2023, Vol. 18 Issue 7, p1-16, 16p
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7 . Academic Journal
Structural basis of the mycobacterial stress-response RNA polymerase auto-inhibition via oligomerization.
저자
by
Morichaud, Zakia
;
Trapani, Stefano
;
Vishwakarma, Rishi K.
;
Chaloin, Laurent
;
Lionne, Corinne
, et al.
소스
Nature Communications; 1/30/2023, Vol. 14 Issue 1, p1-13, 13p
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7 . Academic Journal
CD73 inhibition by purine cytotoxic nucleoside analogue-based diphosphonates
저자
by
Dumontet, Charles
;
Peyrottes, Suzanne
;
Rabeson, Céline
;
Cros-Perrial, Emeline
;
Géant, Pierre Yves
, et al.
소스
In
European Journal of Medicinal Chemistry
5 September 2018 157:1051-1055
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