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1 . Academic Journal
Remibrutinib, a Novel Bruton Tyrosine Kinase Inhibitor, Exhibits Improved Target Selectivity and Potency in Vitro
저자
by
Pulz, Robert
;
Angst, Daniela
;
Eichlisberger, Denis
;
Hayek, Gisele El
;
Cenni, Bruno
.
소스
In
Multiple Sclerosis and Related Disorders
December 2023 80
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7 . Academic Journal
Efficacy and safety of remibrutinib, a selective potent oral BTK inhibitor, in Sjögren's syndrome: results from a randomised, double-blind, placebo-controlled phase 2 trial.
저자
by
Dörner, Thomas
;
Kaul, Martin
;
Szántó, Antónia
;
Jui-Cheng Tseng
;
Papas, Athena S.
, et al.
소스
Annals of the Rheumatic Diseases; Mar2024, Vol. 83 Issue 3, p360-371, 25p
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7 . Academic Journal
Remibrutinib (LOU064) inhibits neuroinflammation driven by B cells and myeloid cells in preclinical models of multiple sclerosis.
저자
by
Nuesslein-Hildesheim, Barbara
;
Ferrero, Enrico
;
Schmid, Cindy
;
Huck, Catherine
;
Smith, Paul
, et al.
소스
Journal of Neuroinflammation
. 8/26/2023, Vol. 20 Issue 1, p1-12. 12p.
Open Access (BioMed Central)
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7 . Academic Journal
Remibrutinib inhibits hives effector cells stimulated by serum from chronic urticaria patients independently of FcεR1 expression level and omalizumab clinical response.
저자
by
Gimeno, Ramón
;
Ribas‐Llauradó, Clara
;
Pesque, David
;
Andrades, Evelyn
;
Cenni, Bruno
, et al.
소스
Clinical & Translational Allergy
. Mar2023, Vol. 13 Issue 3, p1-11. 11p.
Open Access (Wiley)
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7 . Academic Journal
Ligand-independent Activation of Steroid Receptors: New Roles for Old Players
저자
by
Cenni, Bruno
;
Picard, Didier
.
소스
In
Trends in Endocrinology & Metabolism
1999 10(2):41-46
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4 . Academic Journal
Remibrutinib (LOU064): A selective potent oral BTK inhibitor with promising clinical safety and pharmacodynamics in a randomized phase I trial.
저자
by
Kaul, Martin
;
End, Peter
;
Cabanski, Maciej
;
Schuhler, Carole
;
Jakab, Annamaria
, et al.
소스
CTS: Clinical & Translational Science
. Sep2021, Vol. 14 Issue 5, p1756-1768. 13p.
Open Access (Wiley)
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7 . Academic Journal
Design of Potent and Selective Covalent Inhibitors of Bruton's Tyrosine Kinase Targeting an Inactive Conformation.
저자
by
Pulz, Robert
;
Angst, Daniela
;
Dawson, Janet
;
Gessier, Francois
;
Gutmann, Sascha
, et al.
소스
ACS Medicinal Chemistry Letters; 2019, Vol. 10 Issue 10, p1467-1472, 6p
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7 . Periodical
Discovery of LOU064 (Remibrutinib), a Potent and Highly Selective Covalent Inhibitor of Bruton’s Tyrosine Kinase
저자
by
Angst, Daniela
;
Gessier, François
;
Janser, Philipp
;
Vulpetti, Anna
;
Wälchli, Rudolf
, et al.
소스
Journal of Medicinal Chemistry; May 2020, Vol. 63 Issue: 10 p5102-5118, 17p
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7 . Academic Journal
Endothelial Bmx tyrosine kinase activity is essential for myocardial hypertrophy and remodeling.
저자
by
Holopainen, Tanja
;
Räsänen, Markus
;
Anisimov, Andrey
;
Tuomainen, Tomi
;
Wei Zheng
, et al.
소스
Proceedings of the National Academy of Sciences of the United States of America
. 10/20/2015, Vol. 112 Issue 42, p13063-13068. 6p.
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7 . Academic Journal
BMX and Its Role in Inflammation, Cardiovascular Disease, and Cancer.
저자
by
Cenni, Bruno
;
Gutmann, Sascha
;
Gottar-Guillier, Marie
.
소스
International Reviews of Immunology
. Apr2012, Vol. 31 Issue 2, p166-173. 8p. 2 Diagrams.
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