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1 .
Kinetic and Mechanistic Investigations to Enable a Key Suzuki Coupling for Sotorasib Manufacture─What a Difference a Base Makes
저자
by
James I. Murray
;
Liang Zhang
;
Adam Simon
;
Maria V. Silva Elipe
;
Carolyn S. Wei
, et al.
소스
Organic Process Research & Development
. 27:198-205
Web of Science
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7 .
Development of a Commercial Manufacturing Process for Sotorasib, a First-in-Class KRASG12C Inhibitor
저자
by
Liang Zhang
;
Daniel J. Griffin
;
Matthew G. Beaver
;
Laura E. Blue
;
Christopher J. Borths
, et al.
소스
Organic Process Research & Development
. 26:3115-3125
Web of Science
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7 .
Synthesis of Substituted Pyridines via Formal (3+3) Cycloaddition of Enamines with Unsaturated Aldehydes and Ketones
저자
by
Xi-Jie Dai
;
Paul Krolikowski
;
James I. Murray
;
Carolyn S. Wei
;
Peter K. Dornan
, et al.
소스
The Journal of Organic Chemistry
. 87:8437-8444
Web of Science
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7 .
Effects of Multiple Catalyst Deactivation Pathways and Continuous Ligand Recycling on the Kinetics of Pd-Catalyzed C–N Coupling Reactions
저자
by
Keming Zhu
;
Neil A. Strotman
;
Yi Hsiao
;
Martin D. Eastgate
;
Carolyn S. Wei
, et al.
소스
The Journal of Organic Chemistry
. 84:4653-4660
Web of Science
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7 .
Adventures in Atropisomerism: Total Synthesis of a Complex Active Pharmaceutical Ingredient with Two Chirality Axes
저자
by
Thomas M. Razler
;
Jianji Wang
;
Yi Hsiao
;
Yuping Qiu
;
Thorsten Rosner
, et al.
소스
Organic Letters
. 20:3736-3740
Open Access (OpenAIRE)
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7 .
Development of Robust, Scaleable Catalytic Processes through Fundamental Understanding of Reaction Mechanisms
저자
by
Carolyn S. Wei
;
Yi Hsaio
;
Eric M. Simmons
;
Martin D. Eastgate
.
소스
Topics in Catalysis
. 60:620-630
Web of Science
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6 .
C-H Arylation in the Formation of a Complex Pyrrolopyridine, the Commercial Synthesis of the Potent JAK2 Inhibitor, BMS-911543
저자
by
Richard J. Fox
;
Michael B. Hay
;
Gregory L. Beutner
;
Keming Zhu
;
Carolyn S. Wei
, et al.
소스
The Journal of organic chemistry
. 84(8)
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7 .
Ni-Catalyzed C–H Functionalization in the Formation of a Complex Heterocycle: Synthesis of the Potent JAK2 Inhibitor BMS-911543
저자
by
Jacob Albrecht
;
Dimitri Skliar
;
Richard J. Fox
;
Keming Zhu
;
Kristy Tran
, et al.
소스
The Journal of Organic Chemistry
. 80:6001-6011
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7 .
Development of a scalable palladium-catalyzed α-arylation process for the synthesis of a CGRP antagonist
저자
by
Fanfair Dayne Dustan
;
David K. Leahy
;
Yi Hsiao
;
Carolyn S. Wei
;
Thorsten Rosner
, et al.
소스
Tetrahedron
. 69:5677-5684
Web of Science
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7 .
The Impact of Palladium(II) Reduction Pathways on the Structure and Activity of Palladium(0) Catalysts
저자
by
Srinivas Tummala
;
Geraint Davies
;
Qi Gao
;
Yi Hsiao
;
Omid Soltani
, et al.
소스
Angewandte Chemie
. 125:5934-5938
Full Text (Wiley)
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