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1 . Academic Journal
Discovery and Biological Characterization of (2R,4S)-1â²-Acetyl-N-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethyl}-2-(4-fluoro-2-methylphenyl)-N-methyl-4,4â²-bipiperidine-1-carboxamide as a New Potent and Selective Neurokinin 1 (NK1) Receptor Antagonist Clinical Candidate
저자
by
Romano Di Fabio
;
Giuseppe Alvaro
;
Cristiana Griffante
;
Domenica A. Pizzi
;
Daniele Donati
, et al.
소스
Journal of Medicinal Chemistry
. Feb2011, Vol. 54 Issue 4, p1071-1079. 9p.
Full Text (ACS)
Web of Science
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7 . Academic Journal
Exploration of the Amine Terminus in a Novel Series of 1,2,4-Triazolo-3-yl-azabicyclo[3.1.0]hexanes as Selective Dopamine D3Receptor Antagonists.
저자
by
Fabrizio Micheli
;
Luca Arista
;
Barbara Bertani
;
Simone Braggio
;
Anna Maria Capelli
, et al.
소스
Journal of Medicinal Chemistry
. Oct2010, Vol. 53 Issue 19, p7129-7139. 11p.
Full Text (ACS)
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7 . Academic Journal
1,2,4-Triazolyl Azabicyclo[3.1.0]hexanes: A New Series of Potent and Selective Dopamine D
3
Receptor Antagonists.
저자
by
Fabrizio Micheli
;
Luca Arista
;
Giorgio Bonanomi
;
Frank E. Blaney
;
Simone Braggio
, et al.
소스
Journal of Medicinal Chemistry
. Jan2010, Vol. 53 Issue 1, p374-391. 18p.
Full Text (ACS)
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7 . Academic Journal
Discovery Process and Pharmacological Characterization of 2-(S)-(4-Fluoro-2-methylphenyl)piperazine-1-carboxylic Acid [1-(R)-(3,5-Bis-trifluoromethylphenyl)ethyl]methylamide (Vestipitant) as a Potent, Selective, and Orally Active NK1Receptor Antagonist.
저자
by
Romano Di Fabio
;
Cristiana Griffante
;
Giuseppe Alvaro
;
Giorgio Pentassuglia
;
Domenica A. Pizzi
, et al.
소스
Journal of Medicinal Chemistry
. May2009, Vol. 52 Issue 10, p3238-3247. 10p.
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7 . Academic Journal
Dihydropyrrole[2,3-d]pyridine Derivatives as Novel Corticotropin-Releasing Factor-1 Antagonists: Mapping of the Receptor Binding Pocket by in Silico Docking Studies.
저자
by
Romano Di Fabio
;
Roberto Arban
;
Giovanni Bernasconi
;
Simone Braggio
;
Frank E. Blaney
, et al.
소스
Journal of Medicinal Chemistry
. Nov2008, Vol. 51 Issue 22, p7273-7286. 14p.
Full Text (ACS)
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7 . Academic Journal
Design, Synthesis, and Biological Evaluation of Novel Aminobisphosphonates Possessing an in Vivo Antitumor Activity Through a γδ-T Lymphocytes-Mediated Activation Mechanism.
저자
by
Daniele Simoni
;
Nicola Gebbia
;
Francesco Paolo Invidiata
;
Marco Eleopra
;
Paolo Marchetti
, et al.
소스
Journal of Medicinal Chemistry
. Oct2008, Vol. 51 Issue 21, p6800-6807. 8p.
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7 . Academic Journal
Iodine-Mediated Cyclization of (4R,5R)-4,5-Diamino-N,N′-bis[(1S)-1-phenylethyl]-1,7-octadiene – A Stereoselective Route to 2,5-Diazabicyclo[2.2.1]heptanes.
저자
by
Claudio Fiorelli
;
Carla Marchioro
;
Gianluca Martelli
;
Magda Monari
;
Diego Savoia
.
소스
European Journal of Organic Chemistry; Sep2005, Vol. 2005 Issue 18, p3987-3993, 7p
Web of Science
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7 .
Identification, biological characterization and pharmacophoric analysis of a new potent and selective NK1 receptor antagonist clinical candidate
저자
by
Alessandro Poffe
;
Simone Spada
;
Carla Marchioro
;
Mauro Corsi
;
Romano Di Fabio
, et al.
소스
Bioorganic & Medicinal Chemistry
. 21:6264-6273
Web of Science
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7 .
Design, synthesis, and biological evaluation of novel aminobisphosphonates possessing an in vivo antitumor activity through a gammadelta-T lymphocytes-mediated activation mechanism
저자
by
Daniele Simoni
;
Aaron Kwaasi
;
Riccardo Baruchello
;
James E. Dunford
;
Carla Marchioro
, et al.
소스
Open Access (OpenAIRE)
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7 .
Synthesis and biological activity of a novel class nicotinic acetylcholine receptors (nAChRs) ligands structurally related to anatoxin-a
저자
by
Daniele Simoni
;
Riccardo Giovannini
;
Paolo Marchetti
;
Giuseppina Barbato
;
Giuseppina Grisolia
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 21:5423-5427
Open Access (OpenAIRE)
Web of Science
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