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1 .
Process Development of the BACE Inhibitors BI 1147560 BS and BI 1181181 MZ
저자
by
Guisheng Li
;
Zhulin Tan
;
Yibo Xu
;
Kanwar P. S. Sidhu
;
Bo Qu
, et al.
소스
Organic Process Research & Development
. 26:3345-3372
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7 .
A Noncoordinating Acid–Base Catalyst for the Mild and Nonreversible tert-Butylation of Alcohols and Phenols
저자
by
Suttipol Radomkit
;
Daniel R. Fandrick
;
Stefan Braith
;
Chris H. Senanayake
;
Arindom Chatterjee
, et al.
소스
The Journal of Organic Chemistry
. 86:4877-4882
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7 .
Sulfone-Mediated SNAr Reaction as a Powerful Tool for the Synthesis of 4-Quinolinyl Ethers and More—Application to the Synthesis of HCV NS3/4a Protease Inhibitor BI 201420
저자
by
Heewon Lee
;
Nelu Grinberg
;
Nitinchandra D. Patel
;
Andrew Ye
;
Azad Hossain
, et al.
소스
The Journal of Organic Chemistry
. 85:8339-8351
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7 . Academic Journal
PAT Applicationin the Expedited Development of aThree-Step, One-Stage Synthesis of the Dipeptide Intermediate of HCVProtease Inhibitor Faldaprevir.
저자
by
Nizar Haddad
;
Bo Qu
;
Heewon Lee
;
Jon Lorenz
;
Rich Varsolona
, et al.
소스
Organic Process Research & Development; Jan2015, Vol. 19 Issue 1, p132-138, 7p
Full Text (ACS)
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7 .
Atom-Economical Cross-Coupling of Internal and Terminal Alkynes to Access 1,3-Enynes
저자
by
Omar Apolinar
;
Daniel R. Fandrick
;
Rei Matsuura
;
Jinhua Song
;
Mingyu Liu
, et al.
소스
J Am Chem Soc
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7 .
Rational Design of New Dihydrobenzooxophosphole-Based Lewis Base Organocatalysts
저자
by
Jinghua J. Song
;
Anjan Saha
;
Zhengxu S. Han
;
Mac G. Schumer
;
Bo Qu
, et al.
소스
Synlett
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7 .
Safety Assessment of Benzyne Generation from a Silyl Triflate Precursor
저자
by
Carl A. Busacca
;
Jose M. Medina
;
Ivan Volchkov
;
Max Sarvestani
;
Andrew V. Kelleghan
, et al.
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Org Lett
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7 .
Enantioselective Arylation of Oxindoles Using Modified BI-DIME Ligands
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by
Christian A. Malapit
;
Heewon Lee
;
Sonia Rodriguez
;
Hari P. R. Mangunuru
;
Carl A. Busacca
, et al.
소스
Synthesis
. 50:4435-4443
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7 .
Potent and selective CC chemokine receptor 1 antagonists labeled with carbon-13, carbon-14, and tritium
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by
Maxim Cheveliakov
;
Matt Hrapchak
;
Carl A. Busacca
;
Jonathan T. Reeves
;
Bachir Latli
, et al.
소스
Journal of Labelled Compounds and Radiopharmaceuticals
. 61:764-772
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7 .
The Guareschi–Thorpe Cyclization Revisited – An Efficient Synthesis of Substituted 2,6-Dihydroxypyridines and 2,6-Dichloropyridines
저자
by
Chris H. Senanayake
;
Carl A. Busacca
;
Diana C. Reeves
;
Jinghua Xu
;
Xingzhong Zeng
, et al.
소스
Synlett
. 29:1455-1460
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