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1 . Periodical
Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii: From Screening Impurity to In VivoEfficacy
저자
by
Skudlarek, Jason W.
;
Cooke, Andrew J.
;
Mitchell, Helen J.
;
Babaoglu, Kerim
;
Shaw, Anthony W.
, et al.
소스
Journal of Medicinal Chemistry; September 2024, Vol. 67 Issue: 17 p15620-15675, 56p
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7 . Academic Journal
Invention of MK-7845, a SARS-CoV‑2 3CL Protease Inhibitor Employing a Novel Difluorinated Glutamine Mimic.
저자
by
Shurtleff, Valerie W.
;
Layton, Mark E.
;
Parish, Craig A.
;
Perkins, James J.
;
Schreier, John D.
, et al.
소스
Journal of Medicinal Chemistry; 3/14/2024, Vol. 67 Issue 5, p3935-3958, 24p
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7 . Academic Journal
Cerastecins inhibit membrane lipooligosaccharide transport in drug-resistant Acinetobacter baumannii
저자
by
Wang, Hao
;
Ishchenko, Andrii
;
Skudlarek, Jason
;
Shen, Pamela
;
Dzhekieva, Liudmila
, et al.
소스
Nature Microbiology
. 9(5):1244-1255
Web of Science
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7 . Academic Journal
Discovery of novel N-1 substituted pyrazolopyrimidinones as potent, selective PDE2 inhibitors
저자
by
Morriello, Gregori J.
;
Dwyer, Michael P.
;
Chen, Yili
;
Ginetti, Anthony T.
;
Xu, Shimin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 July 2021 44
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7 . Academic Journal
The identification of a novel lead class for phosphodiesterase 2 inhibition by fragment-based drug design
저자
by
Forster, Ashley B.
;
Abeywickrema, Pravien
;
Bunda, Jaime
;
Cox, Christopher D.
;
Cabalu, Tamara D.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2017 27(23):5167-5171
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7 . Academic Journal
Design, synthesis and SAR of substituted indoles as selective TrkA inhibitors
저자
by
Hurzy, Danielle M.
;
Henze, Darrell A.
;
Cabalu, Tamara D.
;
Narayan, Kartik
;
Heller, Amanda
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 June 2017 27(12):2695-2701
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7 . Academic Journal
Investigation of orexin-2 selective receptor antagonists: Structural modifications resulting in dual orexin receptor antagonists
저자
by
Skudlarek, Jason W.
;
DiMarco, Christina N.
;
Babaoglu, Kerim
;
Roecker, Anthony J.
;
Bruno, Joseph G.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 March 2017 27(6):1364-1370
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7 . Academic Journal
Discovery of highly potent and selective orexin 1 receptor antagonists (1-SORAs) suitable for in vivo interrogation of orexin 1 receptor pharmacology
저자
by
Stump, Craig A.
;
Cooke, Andrew J.
;
Bruno, Joseph
;
Cabalu, Tamara D.
;
Gotter, Anthony L.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2016 26(23):5809-5814
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7 . Academic Journal
Discovery of diazepane amide DORAs and 2-SORAs enabled by exploration of isosteric quinazoline replacements
저자
by
Roecker, Anthony J.
;
Mercer, Swati P.
;
Bergman, Jeffrey M.
;
Gilbert, Kevin F.
;
Kuduk, Scott D.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 November 2015 25(21):4992-4999
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7 . Academic Journal
Identification of MK-8133: An orexin-2 selective receptor antagonist with favorable development properties
저자
by
Kuduk, Scott D.
;
Skudlarek, Jason W.
;
DiMarco, Christina N.
;
Bruno, Joseph G.
;
Pausch, Mark H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 June 2015 25(12):2488-2492
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