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1 . Periodical
Chemoproteomic discovery of a covalent allosteric inhibitor of WRN helicase
저자
by
Baltgalvis, Kristen A.
;
Lamb, Kelsey N.
;
Symons, Kent T.
;
Wu, Chu-Chiao
;
Hoffman, Melissa A.
, et al.
소스
Nature; May 2024, Vol. 629 Issue: 8011 p435-442, 8p
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7 . Academic Journal
An efficient one-pot construction of substituted pyrimidinones
저자
by
Lu, Yuelie
;
Xiang, Tingjian
;
Bartberger, Michael D.
;
Bernard, Charles
;
Bostick, Tracy
, et al.
소스
In
Tetrahedron
2006 62(50):11714-11723
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7 . Academic Journal
Tryptase activates peripheral blood mononuclear cells causing the synthesis and release of TNF-α, IL-6 and IL-1β: possible relevance to multiple sclerosis
저자
by
Malamud, Vivian
;
Vaaknin, Ady
;
Abramsky, Oded
;
Mor, Michal
;
Burgess, Laurence E.
, et al.
소스
In
Journal of Neuroimmunology
2003 138(1):115-122
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7 . Academic Journal
Strategies for ansamycin antibiotics. asymmetric synthesis of the C(3)–C(21) subunit of herbimycin A
저자
by
Martin, Stephen F.
;
Limberakis, Chris
;
Burgess, Laurence E.
;
Hartmann, Michael
.
소스
In
Tetrahedron
1999 55(12):3561-3572
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6 . Academic Journal
Identification of the Clinical Development Candidate MRTX849, a Covalent KRAS
G12C
Inhibitor for the Treatment of Cancer.
저자
by
Fell, Jay B.
;
Fischer, John P.
;
Baer, Brian R.
;
Blake, James F.
;
Bouhana, Karyn
, et al.
소스
Journal of Medicinal Chemistry; 7/9/2020, Vol. 63 Issue 13, p6679-6693, 15p
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7 . Periodical
Identification of the Clinical Development Candidate MRTX849, a Covalent KRASG12CInhibitor for the Treatment of Cancer
저자
by
Fell, Jay B.
;
Fischer, John P.
;
Baer, Brian R.
;
Blake, James F.
;
Bouhana, Karyn
, et al.
소스
Journal of Medicinal Chemistry; July 2020, Vol. 63 Issue: 13 p6679-6693, 15p
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7 . Academic Journal
Tetrazole and ester substituted tetrahydoquinoxalines as potent cholesteryl ester transfer protein inhibitors
저자
by
Eary, C. Todd
;
Jones, Zachary S.
;
Groneberg, Robert D.
;
Burgess, Laurence E.
;
Mareska, David A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(9):2608-2613
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7 . Academic Journal
Synthesis of spirolactams and spiropiperidines as CCR4 receptor antagonists
저자
by
Hansen, Joshua D.
;
Newhouse, Bradley J.
;
Allen, Shelley
;
Anderson, Aaron
;
Eary, Todd
, et al.
소스
In
Tetrahedron Letters
2006 47(1):69-72
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7 . Academic Journal
Racemic and chiral lactams as potent, selective and functionally active CCR4 antagonists
저자
by
Newhouse, Bradley
;
Allen, Shelley
;
Fauber, Benjamin
;
Anderson, Aaron S.
;
Eary, C. Todd
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2004 14(22):5537-5542
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7 . Academic Journal
Discovery and SAR of trisubstituted thiazolidinones as CCR4 antagonists
저자
by
Allen, Shelley
;
Newhouse, Bradley
;
Anderson, Aaron S.
;
Fauber, Benjamin
;
Allen, Andrew
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2004 14(7):1619-1624
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