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1 . Academic Journal
Regulation of inositol 5-phosphatase activity by the C2 domain of SHIP1 and SHIP2
저자
by
Bradshaw, William J.
;
Kennedy, Emma C.
;
Moreira, Tiago
;
Smith, Luke A.
;
Chalk, Rod
, et al.
소스
In
Structure
4 April 2024 32(4):453-466
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7 . Academic Journal
Luminescence-based complementation assay to assess target engagement and cell permeability of glycolate oxidase (HAO1) inhibitors
저자
by
Mackinnon, Sabrina R.
;
Zarganes-Tzitzikas, Tryfon
;
Adams, Cassandra J.
;
Brennan, Paul E.
;
Yue, Wyatt W.
.
소스
In
Biochimie
August 2024
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7 . Academic Journal
Discovery of FERM domain protein–protein interaction inhibitors for MSN and CD44 as a potential therapeutic approach for Alzheimer’s disease
저자
by
Du, Yuhong
;
Bradshaw, William J.
;
Leisner, Tina M.
;
Annor-Gyamfi, Joel K.
;
Qian, Kun
, et al.
소스
In
Journal of Biological Chemistry
December 2023 299(12)
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7 . Academic Journal
The X-linked histone demethylases KDM5C and KDM6A as regulators of T cell-driven autoimmunity in the central nervous system
저자
by
Fazazi, Mohamed Reda
;
Ruda, Gian Filippo
;
Brennan, Paul E.
;
Rangachari, Manu
.
소스
In
Brain Research Bulletin
1 October 2023 202
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6 . Academic Journal
C8-substituted pyrido[3,4-d]pyrimidin-4(3H)-ones: Studies towards the identification of potent, cell penetrant Jumonji C domain containing histone lysine demethylase 4 subfamily (KDM4) inhibitors, compound profiling in cell-based target engagement assays
저자
by
Le Bihan, Yann-Vaï
;
Lanigan, Rachel M.
;
Atrash, Butrus
;
McLaughlin, Mark G.
;
Velupillai, Srikannathasan
, et al.
소스
In
European Journal of Medicinal Chemistry
1 September 2019 177:316-337
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7 . Academic Journal
Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2
저자
by
Moustakim, Moses
;
Riedel, Kerstin
;
Schuller, Marion
;
Gehring, Andrè P.
;
Monteiro, Octovia P.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 July 2018 26(11):2965-2972
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7 . Academic Journal
Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells
저자
by
Tumber, Anthony
;
Nuzzi, Andrea
;
Hookway, Edward S.
;
Hatch, Stephanie B.
;
Velupillai, Srikannathasan
, et al.
소스
In
Cell Chemical Biology
16 March 2017 24(3):371-380
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7 . Academic Journal
Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist.
저자
by
Balıkçı, Esra
;
Marques, Anne-Sophie M. C.
;
Bauer, Ludwig G.
;
Seupel, Raina
;
Bennett, James
, et al.
소스
Journal of Medicinal Chemistry; 5/9/2024, Vol. 67 Issue 9, p7245-7259, 15p
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7 . Academic Journal
Development of chemical probes for the bromodomains of BRD7 and BRD9
저자
by
Clark, Peter G.K.
;
Dixon, Darren J.
;
Brennan, Paul E.
.
소스
In
Drug Discovery Today: Technologies
March 2016 19:73-80
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5 . Periodical
Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist
저자
by
Balikc¸i, Esra
;
Marques, Anne-Sophie M. C.
;
Bauer, Ludwig G.
;
Seupel, Raina
;
Bennett, James
, et al.
소스
Journal of Medicinal Chemistry; May 2024, Vol. 67 Issue: 9 p7245-7259, 15p
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