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1 . Academic Journal
Design, synthesis and biological evaluation of 2,3-dihydroimidazo[2,1-b]thiazoles as dual EGFR and IGF1R inhibitors
저자
by
Gadekar, Pradip K.
;
Urunkar, Ganesh
;
Roychowdhury, Abhijit
;
Sharma, Rajiv
;
Bose, Julie
, et al.
소스
In
Bioorganic Chemistry
October 2021 115
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7 . Academic Journal
Cyclopentyl-pyrimidine based analogues as novel and potent IGF-1R inhibitor
저자
by
Aware, Valmik
;
Gaikwad, Nitin
;
Chavan, Sambhaji
;
Manohar, Sonal
;
Bose, Julie
, et al.
소스
In
European Journal of Medicinal Chemistry
6 March 2015 92:246-256
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7 . Academic Journal
Synthesis and evaluation of cyclohexane carboxylic acid head group containing isoxazole and thiazole analogs as DGAT1 inhibitors
저자
by
Kandre, Shivaji
;
Bhagat, Pundlik Rambhau
;
Kumar Reddy, M. Mahesh
;
Dalal, Roda
;
Dixit, Amol
, et al.
소스
In
European Journal of Medicinal Chemistry
22 May 2014 79:203-215
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7 . Academic Journal
A fluorinated analog of ISO-1 blocks the recognition and biological function of MIF and is orally efficacious in a murine model of colitis
저자
by
Dagia, Nilesh M.
;
Kamath, Divya V.
;
Bhatt, Pooja
;
Gupte, Ravindra D.
;
Dadarkar, Shruta S.
, et al.
소스
In
European Journal of Pharmacology
2009 607(1):201-212
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7 . Academic Journal
Discovery of thiazolyl-phthalazinone acetamides as potent glucose uptake activators via high-throughput screening
저자
by
Agrawal, Madhavi
;
Kharkar, Prashant
;
Moghe, Sonali
;
Mahajan, Tushar
;
Deka, Vaishali
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 October 2013 23(20):5740-5743
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7 . Academic Journal
P7170: A Novel Molecule with Unique Profile of mTORC1/C2 and Activin Receptor-like Kinase 1 Inhibition Leading to Antitumor and Antiangiogenic Activity
저자
by
Jalota-Badhwar, Archana
;
Bhatia, Dimple R.
;
Boreddy, Srinivas
;
Joshi, Asavari
;
Venkatraman, Magesh
, et al.
소스
MOLECULAR CANCER THERAPEUTICS
; MAY 2015, 14 5, p1095-p1106, 12p.
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7 . Academic Journal
P7170, a novel inhibitor of mTORC1/mTORC2 and Activin receptor-like Kinase 1 (ALK1) inhibits the growth of non small cell lung cancer
저자
by
Venkatesha, Venkatasubbaiah A.
;
Joshi, Asavari
;
Venkataraman, Magesh
;
Sonawane, Vinay
;
Bhatia, Dimple
, et al.
소스
MOLECULAR CANCER
; DEC 2 2014, 13 p259 11p.
Open Access (BioMed Central)
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7 . Academic Journal
P7170, a novel inhibitor of phosphoinositide 3-kinase (PI3K)-mammalian target of Rapamycin (mTOR) and activin receptor-like kinase 1 (ALK1) as a new therapeutic option for Kras mutated non small cell lung cancer (NSCLC)
저자
by
Agarwal, Veena R.
;
Joshi, Asavari
;
Venkataraman, Magesh
;
Bhatia, Dimple
;
Bose, Julie
, et al.
소스
CANCER RESEARCH
; APR 15 2012, 72 2p. Supplement: 8
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7 . Academic Journal
P7170: A potent and oral phosphoinositide 3-kinase (PI3K)-mammalian target of rapamycin (mTOR) and activin receptor-like kinase 1 (ALK1) inhibitor with anti-tumor and anti-angiogenic activity
저자
by
Agarwal, Veena R.
;
Joshi, Asavari
;
Venkataraman, Magesh
;
Desai, Nikesh
;
Bhatia, Dimple
, et al.
소스
CANCER RESEARCH
; APR 15 2012, 72 2p. Supplement: 8
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7 . Academic Journal
P11187, a Potent and Novel GPR40 Agonist Potentiates Glucose-Stimulated Insulin Secretion, and Improves Glucose Tolerance in Rodent Models of Type 2 Diabetes
저자
by
Anupindi, Raghuram
;
Dixit, Amol
;
Deshmukh, Nitin
;
Gaikwad, Parikshit
;
Patil, Mohan
, et al.
소스
DIABETES
; JUN 2014, 63 pA456-pA456, 1p. Supplement: 1
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