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1 . Academic Journal
C8-substituted pyrido[3,4-d]pyrimidin-4(3H)-ones: Studies towards the identification of potent, cell penetrant Jumonji C domain containing histone lysine demethylase 4 subfamily (KDM4) inhibitors, compound profiling in cell-based target engagement assays
저자
by
Le Bihan, Yann-Vaï
;
Lanigan, Rachel M.
;
Atrash, Butrus
;
McLaughlin, Mark G.
;
Velupillai, Srikannathasan
, et al.
소스
In
European Journal of Medicinal Chemistry
1 September 2019 177:316-337
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7 . Academic Journal
Combining Mutational Signatures, Clonal Fitness, and Drug Affinity to Define Drug-Specific Resistance Mutations in Cancer
저자
by
Kaserer, Teresa
;
Blagg, Julian
.
소스
In
Cell Chemical Biology
15 November 2018 25(11):1359-1371
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4 . Academic Journal
Microfluidic Mobility Shift Assay for Real-Time Analysis of Peptide N-Palmitoylation
저자
by
Lanyon-Hogg, Thomas
;
Patel, Neki V.
;
Ritzefeld, Markus
;
Boxall, Katherine J.
;
Burke, Rosemary
, et al.
소스
In
SLAS Discovery
April 2017 22(4):418-424
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7 . Academic Journal
Design, Synthesis, and Evaluation of Inhibitors of Hedgehog Acyltransferase.
저자
by
Ritzefeld, Markus
;
Zhang, Leran
;
Xiao, Zhangping
;
Andrei, Sebastian A.
;
Boyd, Olivia
, et al.
소스
Journal of Medicinal Chemistry; 1/25/2024, Vol. 67 Issue 2, p1061-1078, 18p
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7 . Academic Journal
Chemical biology approaches to target validation in cancer
저자
by
Blagg, Julian
;
Workman, Paul
.
소스
In
Current Opinion in Pharmacology
August 2014 17:87-100
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4 . Academic Journal
Benzimidazole inhibitors of the protein kinase CHK2: Clarification of the binding mode by flexible side chain docking and protein–ligand crystallography
저자
by
Matijssen, Cornelis
;
Silva-Santisteban, M. Cris
;
Westwood, Isaac M.
;
Siddique, Samerene
;
Choi, Vanessa
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 November 2012 20(22):6630-6639
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7 . Academic Journal
Designing drugs for the treatment of female sexual dysfunction
저자
by
Brown, Alan D.
;
Blagg, Julian
;
Reynolds, David S.
.
소스
In
Drug Discovery Today
2007 12(17):757-766
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5 . Academic Journal
Discovery of potent and selective CDK8 inhibitors from an HSP90 pharmacophore
저자
by
Schiemann, Kai
;
Mallinger, Aurélie
;
Wienke, Dirk
;
Esdar, Christina
;
Poeschke, Oliver
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 March 2016 26(5):1443-1451
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7 . Academic Journal
7-(Pyrazol-4-yl)-3H-imidazo[4,5-b]pyridine-based derivatives for kinase inhibition: Co-crystallisation studies with Aurora-A reveal distinct differences in the orientation of the pyrazole N1-substituent
저자
by
Bavetsias, Vassilios
;
Pérez-Fuertes, Yolanda
;
McIntyre, Patrick J.
;
Atrash, Butrus
;
Kosmopoulou, Magda
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2015 25(19):4203-4209
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7 . Academic Journal
Pyrimido[4,5- d]azepines as potent and selective 5-HT 2C receptor agonists: Design, synthesis, and evaluation of PF-3246799 as a treatment for urinary incontinence
저자
by
Andrews, Mark D.
;
Fish, Paul V.
;
Blagg, Julian
;
Brabham, Tiffini K.
;
Brennan, Paul E.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(9):2715-2720
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