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1 . Academic Journal
Discovery of brain permeable 2-Azabicyclo[2.2.2]octane sulfonamides as a novel class of presenilin-1 selective γ-secretase inhibitors
저자
by
Narlawar, Rajeshwar
;
Serneels, Lutgarde
;
Gaffric, Celia
;
Gijsen, Harrie J.M.
;
De Strooper, Bart
, et al.
소스
In
European Journal of Medicinal Chemistry
15 November 2023 260
Full Text (ScienceDirect)
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7 . Academic Journal
Selective inhibitors of the PSEN1–gamma-secretase complex
저자
by
Serneels, Lutgarde
;
Narlawar, Rajeshwar
;
Perez-Benito, Laura
;
Municoy, Marti
;
Guallar, Victor
, et al.
소스
In
Journal of Biological Chemistry
June 2023 299(6)
Full Text (ScienceDirect)
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7 . Academic Journal
Synthesis and inhibitory activities at mGluRs of 3-alkylated and N-alkylated cyclopentyl-glutamate analogues
저자
by
Ung, Alison T.
;
Pyne, Stephen G.
;
Bischoff, François
;
Lesage, Anne S.J.
;
Skelton, Brian W.
, et al.
소스
In
Tetrahedron
25 March 2013 69(12):2577-2587
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7 . Academic Journal
Synthesis and antagonist activities of 4-aryl-substituted conformationally restricted cyclopentenyl and cyclopentanyl-glutamate analogues
저자
by
Ung, Alison T.
;
Pyne, Stephen G.
;
Batenburg-Nguyen, Uta
;
Davis, Andrew S.
;
Sherif, Azlifa
, et al.
소스
In
Tetrahedron
2005 61(7):1803-1812
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7 . Academic Journal
JNJ16259685, a highly potent, selective and systemically active mGlu1 receptor antagonist
저자
by
Lavreysen, Hilde
;
Wouters, Ria
;
Bischoff, François
;
Nóbrega Pereira, Sandrina
;
Langlois, Xavier
, et al.
소스
In
Neuropharmacology
2004 47(7):961-972
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7 . Academic Journal
Synthesis and characterization of two pet radioligands for the metabotropic glutamate 1 (mGlu1) receptor.
저자
by
Huang, Yiyun
;
Narendran, Rajesh
;
Bischoff, Francois
;
Guo, Ningning
;
Bae, Sung A.
, et al.
소스
Synapse
. Dec2012, Vol. 66 Issue 12, p1002-1014. 13p.
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7 . Academic Journal
Design and Synthesis ofa Novel Series of BicyclicHeterocycles As Potent γ-Secretase Modulators.
저자
by
Bischoff, Francois
;
Berthelot, Didier
;
De Cleyn, Michel
;
Macdonald, Gregor
;
Minne, Garrett
, et al.
소스
Journal of Medicinal Chemistry
. Vol. 55 Issue 21, p9089-9106. 18p.
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7 . Academic Journal
Extracellular interface between APP and Nicastrin regulates Aβ length and response to γ‐secretase modulators.
저자
by
Petit, Dieter
;
Hitzenberger, Manuel
;
Lismont, Sam
;
Zoltowska, Katarzyna Marta
;
Ryan, Natalie S
, et al.
소스
EMBO Journal
. 6/17/2019, Vol. 38 Issue 12, pN.PAG-N.PAG. 1p. 3 Diagrams, 4 Graphs.
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7 . Academic Journal
Synthesis and Pharmacological Characterization of Two Novel, Brain Penetrating P2X(7) Antagonists
저자
by
Letavic, Michael A.
;
Lord, Brian
;
Bischoff, Francois
;
Hawryluk, Natalie A.
;
Pieters, Serge
, et al.
소스
ACS MEDICINAL CHEMISTRY LETTERS
; APR 2013, 4 4, p419-p422, 4p.
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7 . Academic Journal
2-amino-3,4-dihydroquinazolines as inhibitors of BACE-1 (beta-site APP cleaving enzyme): Use of structure based design to convert a micromolar hit into a nanomolar lead
저자
by
Baxter, Ellen W.
;
Conway, Kelly A.
;
Kennis, Ludo
;
Bischoff, Francois
;
Mercken, Marc H.
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; SEP 6 2007, 50 18, p4261-p4264, 4p.
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