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1 . Academic Journal
Calculation and application of activity discriminants in lead optimization
저자
by
Luo, Xincai
;
Krumrine, Jennifer R.
;
Shenvi, Ashok B.
;
Pierson, M. Edward
;
Bernstein, Peter R.
.
소스
In
Journal of Molecular Graphics and Modelling
2010 29(3):372-381
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7 . Academic Journal
Naphtho[2,1- b][1,5] and [1,2- f][1,4]oxazocines as selective NK 1 antagonists
저자
by
Ohnmacht, Cyrus J.
;
Albert, Jeffrey S.
;
Bernstein, Peter R.
;
Rumsey, William L.
;
Masek, Brian B.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2004 12(10):2653-2669
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7 . Periodical
Pharmacophore-Based Design of Phenyl-[hydroxycyclohexyl] Cycloalkyl-Carboxamide Mitofusin Activators with Improved Neuronal Activity
저자
by
Dang, Xiawei
;
Williams, Sidney B.
;
Devanathan, Sriram
;
Franco, Antonietta
;
Fu, Lijun
, et al.
소스
Journal of Medicinal Chemistry; September 2021, Vol. 64 Issue: 17 p12506-12524, 19p
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7 . Academic Journal
Discovery of 6‑Phenylhexanamide Derivatives as Potent Stereoselective Mitofusin Activators for the Treatment of Mitochondrial Diseases.
저자
by
Dang, Xiawei
;
Zhang, Lihong
;
Franco, Antonietta
;
Li, Jiajia
;
Rocha, Agostinho G.
, et al.
소스
Journal of Medicinal Chemistry; 7/9/2020, Vol. 63 Issue 13, p7033-7051, 19p
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7 . Periodical
Discovery of a Potent and Selective PI3Kδ Inhibitor (S)-2,4-Diamino-6-((1-(7-fluoro-1-(4-fluorophenyl)-4-oxo-3-phenyl-4H-quinolizin-2-yl)ethyl)amino)pyrimidine-5-carbonitrile with Improved Pharmacokinetic Profile and Superior Efficacy in Hematological Cancer Models
저자
by
Shukla, Manojkumar R.
;
Patra, Sukanya
;
Verma, Mahip
;
Sadasivam, Gayathri
;
Jana, Nirmal
, et al.
소스
Journal of Medicinal Chemistry; December 2020, Vol. 63 Issue: 23 p14700-14723, 24p
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7 . Academic Journal
Discovery of isoquinolinone and naphthyridinone-based inhibitors of poly (ADP-ribose) polymerase-1 (PARP1) as anticancer agents: Structure activity relationship and preclinical characterization
저자
by
Karche, Navnath P.
;
Bhonde, Mandar
;
Sinha, Neelima
;
Jana, Gourhari
;
Kukreja, Gagan
, et al.
소스
BIOORGANIC & MEDICINAL CHEMISTRY
; DEC 15 2020, 28 24, p115819 17p.
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7 . Academic Journal
Discovery of a Potent and Selective PI3K delta Inhibitor (S)-2,4-Diamino-6-((1-(7-fluoro-1-(4-fluorophenyl)-4-oxo-3-phenyl-4H-quinolizin-2-yl)ethyl)amino)pyrimidine-5-carbonitrile with Improved Pharmacokinetic Profile and Superior Efficacy in Hematological Cancer Models
저자
by
Shukla, Manojkumar R.
;
Patra, Sukanya
;
Verma, Mahip
;
Sadasivam, Gayathri
;
Jana, Nirmal
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; DEC 10 2020, 63 23, p14700-p14723, 24p.
Full Text (ACS)
Scopus
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7 . Academic Journal
Discovery of novel, orally active dual NK 1/NK 2 antagonists
저자
by
Bernstein, Peter R.
;
Aharony, David
;
Albert, Jeffrey S.
;
Andisik, Donald
;
Barthlow, Herbert G.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2001 11(20):2769-2773
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7 . Academic Journal
Discovery of Spirofused Piperazineand Diazepane Amidesas Selective Histamine-3 Antagonists with in Vivo Efficacyin a Mouse Model of Cognition.
저자
by
Brown, Dean G.
;
Bernstein, Peter R.
;
Griffin, Andrew
;
Wesolowski, Steve
;
Labrecque, Denis
, et al.
소스
Journal of Medicinal Chemistry
. Feb2014, Vol. 57 Issue 3, p733-758. 26p.
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7 . Academic Journal
Naphtho[2,1-b][1,5] and [1,2-f][1,4]oxazocines as selective NK
1
antagonists
저자
by
Ohnmacht, Cyrus J.
;
Albert, Jeffrey S.
;
Bernstein, Peter R.
;
Rumsey, William L.
;
Masek, Brian B.
, et al.
소스
Bioorganic & Medicinal Chemistry
. May2004, Vol. 12 Issue 10, p2653. 17p.
Full Text (ScienceDirect)
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