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1 . Academic Journal
Low-data interpretable deep learning prediction of antibody viscosity using a biophysically meaningful representation.
저자
by
Rai, Brajesh K.
;
Apgar, James R.
;
Bennett, Eric M.
.
소스
Scientific Reports
. 2/20/2023, Vol. 13 Issue 1, p1-13. 13p.
Web of Science
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5 . Academic Journal
Reduction of therapeutic antibody self-association using yeast-display selections and machine learning.
저자
by
Makowski, Emily K.
;
Chen, Hongwei
;
Lambert, Matthew
;
Bennett, Eric M.
;
Eschmann, Nicole S.
, et al.
소스
mAbs; Jan-Dec2022, Vol. 14 Issue 1, p1-14, 14p
Open Access (T&F)
Web of Science
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7 . Academic Journal
Identification and optimization of indolo[2,3-c]quinoline inhibitors of IRAK4
저자
by
Tumey, L. Nathan
;
Boschelli, Diane H.
;
Bhagirath, Niala
;
Shim, Jaechul
;
Murphy, Elizabeth A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 May 2014 24(9):2066-2072
Full Text (ScienceDirect)
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7 . Academic Journal
Combining random mutagenesis, structure-guided design and next-generation sequencing to mitigate polyreactivity of an anti-IL-21R antibody.
저자
by
Campbell, Sharon M.
;
DeBartolo, Joseph
;
Apgar, James R.
;
Mosyak, Lydia
;
McManus, Virginie
, et al.
소스
mAbs; Jan-Dec 2021, Vol. 13 Issue 1, p1-13, 13p
Open Access (T&F)
Web of Science
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7 . Academic Journal
Identification of pyrimidine derivatives as hSMG-1 inhibitors
저자
by
Gopalsamy, Ariamala
;
Bennett, Eric M.
;
Shi, Mengxiao
;
Zhang, Wei-Guo
;
Bard, Joel
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 November 2012 22(21):6636-6641
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7 . Academic Journal
Modeling and mitigation of high-concentration antibody viscosity through structure-based computer-aided protein design.
저자
by
Apgar, James R.
;
Tam, Amy S. P.
;
Sorm, Rhady
;
Moesta, Sybille
;
King, Amy C.
, et al.
소스
PLoS ONE
. 5/7/2020, Vol. 15 Issue 5, p1-26. 26p.
Web of Science
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7 . Academic Journal
Synthesis of 4-phenoxybenzamide adenine dinucleotide as NAD analogue with inhibitory activity against enoyl-ACP reductase (InhA) of Mycobacterium tuberculosis
저자
by
Bonnac, Laurent
;
Gao, Guang-Yao
;
Chen, Liqiang
;
Felczak, Krzysztof
;
Bennett, Eric M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 August 2007 17(16):4588-4591
Full Text (ScienceDirect)
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7 . Academic Journal
Methylenebis(sulfonamide) linked nicotinamide adenine dinucleotide analogue as an inosine monophosphate dehydrogenase inhibitor
저자
by
Chen, Liqiang
;
Gao, Guangyao
;
Bonnac, Laurent
;
Wilson, Daniel J.
;
Bennett, Eric M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(11):3152-3155
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7 . Academic Journal
PF-06804103, A Site-specific Anti-HER2 Antibody-Drug Conjugate for the Treatment of HER2-expressing Breast, Gastric, and Lung Cancers
저자
by
Graziani, Edmund, I
;
Sung, Matthew
;
Ma, Dangshe
;
Narayanan, Bitha
;
Marquette, Kimberly
, et al.
소스
MOLECULAR CANCER THERAPEUTICS
; OCT 1 2020, 19 10, p2068-p2078, 11p.
Full Text (AACR)
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7 . Academic Journal
AB-Bind: Antibody binding mutational database for computational affinity predictions
저자
by
Sirin, Sarah
;
Apgar, James R.
;
Bennett, Eric M.
;
Keating, Amy E.
.
소스
Protein Science
. Feb 01, 2016 25(2):393-409
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