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1 . Academic Journal
C8-substituted pyrido[3,4-d]pyrimidin-4(3H)-ones: Studies towards the identification of potent, cell penetrant Jumonji C domain containing histone lysine demethylase 4 subfamily (KDM4) inhibitors, compound profiling in cell-based target engagement assays
저자
by
Le Bihan, Yann-Vaï
;
Lanigan, Rachel M.
;
Atrash, Butrus
;
McLaughlin, Mark G.
;
Velupillai, Srikannathasan
, et al.
소스
In
European Journal of Medicinal Chemistry
1 September 2019 177:316-337
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7 . Academic Journal
Synthesis and profiling of a 3-aminopyridin-2-one-based kinase targeted fragment library: Identification of 3-amino-5-(pyridin-4-yl)pyridin-2(1H)-one scaffold for monopolar spindle 1 (MPS1) and Aurora kinases inhibition
저자
by
Fearon, Daren
;
Westwood, Isaac M.
;
van Montfort, Rob L.M.
;
Bayliss, Richard
;
Jones, Keith
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 July 2018 26(11):3021-3029
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7 . Academic Journal
Synthesis of isothiazol-3-one derivatives as inhibitors of histone acetyltransferases (HATs)
저자
by
Gorsuch, Stephen
;
Bavetsias, Vassilios
;
Rowlands, Martin G.
;
Aherne, G. Wynne
;
Workman, Paul
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2009 17(2):467-474
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7 . Academic Journal
Cyclopenta[ g]quinazolinone-based inhibitors of thymidylate synthase targeting α-folate receptor overexpressing tumours: synthetic approaches to 4-{ N-[(6 RS)-2-hydroxymethyl-4-oxo-3,4,7,8-tetrahydro-6 H-cyclopenta[ g]quinazolin-6-yl]- N-(prop-2-ynyl)amino}benzoic acid
저자
by
Bavetsias, Vassilios
;
Henderson, Elisa A.
;
McDonald, Edward
.
소스
In
Tetrahedron
2007 63(7):1537-1543
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5 . Academic Journal
Targeting the α-folate receptor with cyclopenta[ g]quinazoline-based inhibitors of thymidylate synthase
저자
by
Henderson, Elisa A.
;
Bavetsias, Vassilios
;
Theti, Davinder S.
;
Wilson, Stuart C.
;
Clauss, Rainer
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2006 14(14):5020-5042
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7 . Academic Journal
Structure-based design of isoquinoline-5-sulfonamide inhibitors of protein kinase B
저자
by
Collins, Ian
;
Caldwell, John
;
Fonseca, Tatiana
;
Donald, Alastair
;
Bavetsias, Vassilios
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2006 14(4):1255-1273
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7 . Academic Journal
7-(Pyrazol-4-yl)-3H-imidazo[4,5-b]pyridine-based derivatives for kinase inhibition: Co-crystallisation studies with Aurora-A reveal distinct differences in the orientation of the pyrazole N1-substituent
저자
by
Bavetsias, Vassilios
;
Pérez-Fuertes, Yolanda
;
McIntyre, Patrick J.
;
Atrash, Butrus
;
Kosmopoulou, Magda
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2015 25(19):4203-4209
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7 . Academic Journal
CCT245718, a dual FLT3/Aurora A inhibitor overcomes D835Y-mediated resistance to FLT3 inhibitors in acute myeloid leukaemia cells.
저자
by
Tariq, Muhammad Usama
;
Furqan, Muhammad
;
Parveen, Hira
;
Ullah, Rahim
;
Muddassar, Muhammad
, et al.
소스
British Journal of Cancer
. Sep2021, Vol. 125 Issue 7, p966-974. 9p.
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7 . Academic Journal
Structure-based design of imidazo[1,2- a]pyrazine derivatives as selective inhibitors of Aurora-A kinase in cells
저자
by
Bouloc, Nathalie
;
Large, Jonathan M.
;
Kosmopoulou, Magda
;
Sun, Chongbo
;
Faisal, Amir
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(20):5988-5993
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7 . Academic Journal
Microwave-assisted synthesis of 2-aminonicotinic acids by reacting 2-chloronicotinic acid with amines
저자
by
Quevedo, Camilo E.
;
Bavetsias, Vassilios
;
McDonald, Edward
.
소스
In
Tetrahedron Letters
2009 50(21):2481-2483
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