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1 . Academic Journal
1,2,4-Amino-triazine derivatives as pyruvate dehydrogenase kinase inhibitors: Synthesis and pharmacological evaluation
저자
by
Pecoraro, Camilla
;
De Franco, Michele
;
Carbone, Daniela
;
Bassani, Davide
;
Pavan, Matteo
, et al.
소스
In
European Journal of Medicinal Chemistry
5 March 2023 249
Full Text (ScienceDirect)
Web of Science
Scopus
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7 . Periodical
Another string to your bow: machine learning prediction of the pharmacokinetic properties of small molecules
저자
by
Bassani, Davide
;
Parrott, Neil John
;
Manevski, Nenad
;
Zhang, Jitao David
.
소스
Expert Opinion on Drug Discovery; June 2024, Vol. 19 Issue: 6 p683-698, 16p
Web of Science
Scopus
JCR 저널정보
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6 . Academic Journal
Molecular Modeling Unveils the Effective Interaction of B-RAF Inhibitors with Rare B-RAF Insertion Variants.
저자
by
Scaini, Maria Chiara
;
Piccin, Luisa
;
Bassani, Davide
;
Scapinello, Antonio
;
Pellegrini, Stefania
, et al.
소스
International Journal of Molecular Sciences
. Aug2023, Vol. 24 Issue 15, p12285. 15p.
JCR 저널정보
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7 . Academic Journal
Are Two Riboses Better Than One? The Case of the Recognition and Activation of Adenosine Receptors.
저자
by
Gianferrara, Teresa
;
Pavan, Matteo
;
Bassani, Davide
;
Vincenzi, Fabrizio
;
Pasquini, Silvia
, et al.
소스
ChemMedChem; 7/17/2023, Vol. 18 Issue 14, p1-14, 14p
Web of Science
Scopus
JCR 저널정보
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7 . Academic Journal
Past, Present, and Future Perspectives on Computer-Aided Drug Design Methodologies.
저자
by
Bassani, Davide
;
Moro, Stefano
.
소스
Molecules
. May2023, Vol. 28 Issue 9, p3906. 20p.
Web of Science
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4 . Academic Journal
Structural Manipulations of Marine Natural Products Inspire a New Library of 3-Amino-1,2,4-Triazine PDK Inhibitors Endowed with Antitumor Activity in Pancreatic Ductal Adenocarcinoma.
저자
by
Carbone, Daniela
;
De Franco, Michele
;
Pecoraro, Camilla
;
Bassani, Davide
;
Pavan, Matteo
, et al.
소스
Marine Drugs; May2023, Vol. 21 Issue 5, p288, 21p
Web of Science
Scopus
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7 . Academic Journal
Discovery of the 3-Amino-1,2,4-triazine-Based Library as Selective PDK1 Inhibitors with Therapeutic Potential in Highly Aggressive Pancreatic Ductal Adenocarcinoma.
저자
by
Carbone, Daniela
;
De Franco, Michele
;
Pecoraro, Camilla
;
Bassani, Davide
;
Pavan, Matteo
, et al.
소스
International Journal of Molecular Sciences
. Feb2023, Vol. 24 Issue 4, p3679. 25p.
JCR 저널정보
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7 . Academic Journal
"Dual Anta-Inhibitors" of the A 2A Adenosine Receptor and Casein Kinase CK1delta: Synthesis, Biological Evaluation, and Molecular Modeling Studies.
저자
by
Spinaci, Andrea
;
Buccioni, Michela
;
Catarzi, Daniela
;
Cui, Chang
;
Colotta, Vittoria
, et al.
소스
Pharmaceuticals (14248247)
. Feb2023, Vol. 16 Issue 2, p167. 30p.
Web of Science
Scopus
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7 . Academic Journal
SARS-CoV-2 3CL
pro
mutations selected in a VSV-based system confer resistance to nirmatrelvir, ensitrelvir, and GC376.
저자
by
Heilmann, Emmanuel
;
Costacurta, Francesco
;
Moghadasi, Seyed Arad
;
Ye, Chengjin
;
Pavan, Matteo
, et al.
소스
Science Translational Medicine; 1/11/2023, Vol. 15 Issue 678, p1-18, 18p
Web of Science
Scopus
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7 . Academic Journal
Physiologically Based Biopharmaceutics Modeling of Food Effect for Basmisanil: A Retrospective Case Study of the Utility for Formulation Bridging.
저자
by
Belubbi, Tejashree
;
Bassani, Davide
;
Stillhart, Cordula
;
Parrott, Neil
.
소스
Pharmaceutics
. Jan2023, Vol. 15 Issue 1, p191. 11p.
Web of Science
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