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1 .
Discovery and optimization of covalent EGFR T790M/L858R mutant inhibitors
저자
by
Maaike Emmelot
;
Dennis Demont
;
Edwin de Zwart
;
Allard Kaptein
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Bas van de Kar
, et al.
소스
Bioorganicmedicinal chemistry letters
. 52
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7 .
Discovery of quinoline-based irreversible BTK inhibitors
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by
Tjeerd Barf
;
Bart Van Lith
;
Todd Covey
;
Dennis Demont
;
Niels Hoogenboom
, et al.
소스
Bioorganicmedicinal chemistry letters
. 30(14)
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7 .
Direct and two-step bioorthogonal probes for Bruton's tyrosine kinase based on ibrutinib: a comparative study
저자
by
Nora Liu
;
Tjeerd Barf
;
Sascha Hoogendoorn
;
Gijsbert A. van der Marel
;
Bas van de Kar
, et al.
소스
Organic & biomolecular chemistry
Organic and Biomolecular Chemistry, 13(18), 5147-5157
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7 .
Acalabrutinib (ACP-196): A Covalent Bruton Tyrosine Kinase Inhibitor with a Differentiated Selectivity and In Vivo Potency Profile
저자
by
Dennis Demont
;
Roger G. Ulrich
;
Tjeerd Barf
;
Raquel Izumi
;
Allard Kaptein
, et al.
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The Journal of pharmacology and experimental therapeutics
. 363(2)
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7 .
Potency and Selectivity of BTK Inhibitors in Clinical Development for B-Cell Malignancies
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by
Diana Mittag
;
Bas van de Kar
;
Tjeerd Barf
;
Dennis Demont
;
Todd Covey
, et al.
소스
Blood
. 132:1871-1871
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7 .
Novel ATP competitive MK2 inhibitors with potent biochemical and cell-based activity throughout the series
저자
by
Arthur Oubrie
;
Carsten Schultz-Fademrecht
;
Vera de Kimpe
;
Bas van de Kar
;
Tjeerd Barf
, et al.
소스
Bioorganicmedicinal chemistry letters
. 22(1)
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7 .
Discovery of selective and orally available spiro-3-piperidyl ATP-competitive MK2 inhibitors
저자
by
Judith Versteegh
;
Joeri Johannes Petrus De Wit
;
Arthur Oubrie
;
Niels Hoogenboom
;
Tjeerd Barf
, et al.
소스
Bioorganicmedicinal chemistry letters
. 21(12)
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7 .
Structure-based lead identification of ATP-competitive MK2 inhibitors
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by
Judith Versteegh
;
Nicole Seegers
;
Henri Klop
;
Tjeerd Barf
;
Claudia Hofstra
, et al.
소스
Bioorganic & Medicinal Chemistry Letters, 21, 3818-22
Bioorganic & Medicinal Chemistry Letters, 21, 12, pp. 3818-22
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7 .
Abstract 2596: ACP-196: a novel covalent Bruton's tyrosine kinase (Btk) inhibitor with improved selectivity and in vivo target coverage in chronic lymphocytic leukemia (CLL) patients
저자
by
Elena Bibikova
;
Ahmed Hamdy
;
Edwin de Zwart
;
Fanny Krantz
;
Raquel Izumi
, et al.
소스
Cancer Research
. 75:2596-2596
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