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1 . Academic Journal
Drugging the ‘undruggable’. Therapeutic targeting of protein–DNA interactions with the use of computer-aided drug discovery methods
저자
by
Radaeva, Mariia
;
Ton, Anh-Tien
;
Hsing, Michael
;
Ban, Fuqiang
;
Cherkasov, Artem
.
소스
In
Drug Discovery Today
November 2021 26(11):2660-2679
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7 . Academic Journal
Interleukin-10 and Small Molecule SHIP1 Allosteric Regulators Trigger Anti-inflammatory Effects through SHIP1/STAT3 Complexes
저자
by
Chamberlain, Thomas C.
;
Cheung, Sylvia T.
;
Yoon, Jeff S.J.
;
Ming-Lum, Andrew
;
Gardill, Bernd R.
, et al.
소스
In
iScience
21 August 2020 23(8)
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7 . Academic Journal
Computer-aided drug discovery of Myc-Max inhibitors as potential therapeutics for prostate cancer
저자
by
Carabet, Lavinia A.
;
Lallous, Nada
;
Leblanc, Eric
;
Ban, Fuqiang
;
Morin, Helene
, et al.
소스
In
European Journal of Medicinal Chemistry
5 December 2018 160:108-119
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7 . Academic Journal
Small molecule-induced degradation of the full length and V7 truncated variant forms of human androgen receptor
저자
by
Dalal, Kush
;
Morin, Helene
;
Ban, Fuqiang
;
Shepherd, Ashley
;
Fernandez, Michael
, et al.
소스
In
European Journal of Medicinal Chemistry
5 September 2018 157:1164-1173
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7 . Academic Journal
In silico screening of LRRK2 WDR domain inhibitors using deep docking and free energy simulations.
저자
by
Gutkin, Evgeny
;
Gusev, Filipp
;
Gentile, Francesco
;
Ban, Fuqiang
;
Koby, S. Benjamin
, et al.
소스
Chemical Science; 6/21/2024, Vol. 15 Issue 23, p8800-8812, 13p
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7 . Academic Journal
Identification of a Potent Antiandrogen that Targets the BF3 Site of the Androgen Receptor and Inhibits Enzalutamide-Resistant Prostate Cancer
저자
by
Munuganti, Ravi S.N.
;
Hassona, Mohamed D.H.
;
Leblanc, Eric
;
Frewin, Kate
;
Singh, Kriti
, et al.
소스
In
Chemistry & Biology
20 November 2014 21(11):1476-1485
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7 . Academic Journal
Discovery of inhibitors of the mitotic kinase TTK based on N-(3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-acetamides and carboxamides
저자
by
Laufer, Radoslaw
;
Ng, Grace
;
Liu, Yong
;
Patel, Narendra Kumar B.
;
Edwards, Louise G.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 September 2014 22(17):4968-4997
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7 . Academic Journal
A novel class of broad-spectrum active-site-directed 3C-like protease inhibitors with nanomolar antiviral activity against highly immune-evasive SARS-CoV-2 Omicron subvariants.
저자
by
Pérez-Vargas, Jimena
;
Worrall, Liam J.
;
Olmstead, Andrea D.
;
Ton, Anh-Tien
;
Lee, Jaeyong
, et al.
소스
Emerging Microbes & Infections; Dec2023, Vol. 12 Issue 2, p1-17, 17p
Open Access (T&F)
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7 . Academic Journal
Novel Inhibitors of androgen receptor's DNA binding domain identified using an ultra‐large virtual screening.
저자
by
Radaeva, Mariia
;
Morin, Helene
;
Pandey, Mohit
;
Ban, Fuqiang
;
Guo, Maria
, et al.
소스
Molecular Informatics; Aug2023, Vol. 42 Issue 8, p1-7, 7p
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7 . Academic Journal
Large-Scale Virtual Screening for the Discovery of SARS-CoV‑2 Papain-like Protease (PLpro) Non-covalent Inhibitors.
저자
by
Garland, Olivia
;
Ton, Anh-Tien
;
Moradi, Shoeib
;
Smith, Jason R.
;
Kovacic, Suzana
, et al.
소스
Journal of Chemical Information & Modeling; 4/10/2023, Vol. 63 Issue 7, p2158-2169, 12p
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