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1 . Academic Journal
Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii: From Screening Impurity to In Vivo Efficacy.
저자
by
Skudlarek, Jason W.
;
Cooke, Andrew J.
;
Mitchell, Helen J.
;
Babaoglu, Kerim
;
Shaw, Anthony W.
, et al.
소스
Journal of Medicinal Chemistry; 9/12/2024, Vol. 67 Issue 17, p15620-15675, 56p
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7 . Academic Journal
Cerastecins inhibit membrane lipooligosaccharide transport in drug-resistant Acinetobacter baumannii
저자
by
Wang, Hao
;
Ishchenko, Andrii
;
Skudlarek, Jason
;
Shen, Pamela
;
Dzhekieva, Liudmila
, et al.
소스
Nature Microbiology
. 9(5):1244-1255
Web of Science
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7 . Academic Journal
Potent targeted activator of cell kill molecules eliminate cells expressing HIV-1.
저자
by
Balibar, Carl J.
;
Klein, Daniel J.
;
Zamlynny, Beata
;
Diamond, Tracy L.
;
Fang, Zhiyu
, et al.
소스
Science Translational Medicine; 2/22/2023, Vol. 15 Issue 684, p1-12, 12p
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7 . Academic Journal
Topoisomerase Inhibitors Addressing Fluoroquinolone Resistance in Gram-Negative Bacteria.
저자
by
Skepper, Colin K.
;
Armstrong, Duncan
;
Balibar, Carl J.
;
Bauer, Daniel
;
Bellamacina, Cornelia
, et al.
소스
Journal of Medicinal Chemistry; 7/23/2020, Vol. 63 Issue 14, p7773-7816, 44p
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7 . Academic Journal
A small-molecule inhibitor of BamA impervious to efflux and the outer membrane permeability barrier.
저자
by
Hart, Elizabeth M.
;
Mitchell, Angela M.
;
Konovalova, Anna
;
Grabowicz, Marcin
;
Sheng, Jessica
, et al.
소스
Proceedings of the National Academy of Sciences of the United States of America
. 10/22/2019, Vol. 116 Issue 43, p21748-21757. 10p.
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7 . Periodical
Two Distinct Mechanisms of Inhibition of LpxA Acyltransferase Essential for Lipopolysaccharide Biosynthesis
저자
by
Han, Wooseok
;
Ma, Xiaolei
;
Balibar, Carl J.
;
Baxter Rath, Christopher M.
;
Benton, Bret
, et al.
소스
Journal of the American Chemical Society; March 2020, Vol. 142 Issue: 9 p4445-4455, 11p
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7 . Academic Journal
Inhibitor of intramembrane protease RseP blocks the σ
E
response causing lethal accumulation of unfolded outer membrane proteins.
저자
by
Silhavy, Thomas J.
;
Konovalova, Anna
;
Grabowicz, Marcin
;
Rigel, Nathan W.
;
Ricci, Dante P.
, et al.
소스
Proceedings of the National Academy of Sciences of the United States of America
. 7/10/2018, Vol. 115 Issue 28, pE6614-E6621. 8p.
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7 . Academic Journal
Fragment-Based Drug Discovery of Inhibitors of Phosphopantetheine Adenylyltransferase from Gram-Negative Bacteria.
저자
by
Moreau, Robert J.
;
Skepper, Colin K.
;
Appleton, Brent A.
;
Blechschmidt, Anke
;
Balibar, Carl J.
, et al.
소스
Journal of Medicinal Chemistry
. 4/26/2018, Vol. 61 Issue 8, p3309-3324. 16p.
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7 . Academic Journal
Yeast: a microbe with macro-implications to antimicrobial drug discovery
저자
by
Balibar, Carl J.
;
Roemer, Terry
.
소스
Briefings in Functional Genomics
. Mar 01, 2016 15(2):147-154
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4 . Academic Journal
Selective small-molecule inhibition of an RNA structural element.
저자
by
Howe, John A.
;
Wang, Hao
;
Fischmann, Thierry O.
;
Balibar, Carl J.
;
Xiao, Li
, et al.
소스
Nature
. 10/29/2015, Vol. 526 Issue 7575, p672-677. 6p. 1 Black and White Photograph, 4 Diagrams, 2 Charts, 7 Graphs.
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