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1 . Academic Journal
White Paper: Mimetics of Class 2 Tumor Suppressor Proteins as Novel Drug Candidates for Personalized Cancer Therapy
저자
by
Edgar Dahl
;
Sophia Villwock
;
Peter Habenberger
;
Axel Choidas
;
Michael Rose
, et al.
소스
Cancers, Vol 14, Iss 18, p 4386 (2022)
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7 . Academic Journal
Anti-leukemic effect of CDK9 inhibition in T-cell prolymphocytic leukemia
저자
by
Patricia Johansson
;
Laura Dierichs
;
Ludger Klein-Hitpass
;
Anke K. Bergmann
;
Michael Möllmann
, et al.
소스
Therapeutic Advances in Hematology, Vol 11 (2020)
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7 . Academic Journal
Systematic Kinase Inhibitor Profiling Identifies CDK9 as a Synthetic Lethal Target in NUT Midline Carcinoma
저자
by
Johannes Brägelmann
;
Marcel A. Dammert
;
Felix Dietlein
;
Johannes M. Heuckmann
;
Axel Choidas
, et al.
소스
Cell Reports, Vol 20, Iss 12, Pp 2833-2845 (2017)
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7 .
IFNα primes cancer cells for Fusicoccin-induced cell death via 14-3-3 PPI stabilization
저자
by
Blaž Andlovic
;
Geronimo Heilmann
;
Sabrina Ninck
;
Sebastian A. Andrei
;
Federica Centorrino
, et al.
소스
Cell Chemical Biology
.
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7 .
Synthesis, Biological Evaluation, and Binding Mode of a New Class of Oncogenic K‐Ras4b Inhibitors
저자
by
Stephan Jeuken
;
Oleksandr Shkura
;
Marc Röger
;
Victoria Brickau
;
Axel Choidas
, et al.
소스
ChemMedChem
. 17
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7 .
Abstract 416: A novel non-covalent and rapidly reversible proteasome inhibitor for multiple myeloma and various solid cancers
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by
Won-Gyun Ahn
;
Yeejin Jeon
;
Yeong-In Yang
;
Jaeseung Kim
;
Seung-Joo Lee
, et al.
소스
Cancer Research
. 82:416-416
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7 .
Potent anti-leukemic activity of a specific cyclin-dependent kinase 9 inhibitor in mouse models of chronic lymphocytic leukemia
저자
by
Ulrich Lücking
;
Jan Dürig
;
Michael Möllmann
;
Axel Choidas
;
Joachim R. Göthert
, et al.
소스
Oncotarget
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7 .
Identification of an (−)-englerin A analogue, which antagonizes (−)-englerin A at TRPC1/4/5 channels
저자
by
Mathias Christmann
;
Peter Nussbaumer
;
Herbert Waldmann
;
Klaus Dinkel
;
Bert Klebl
, et al.
소스
British Journal of Pharmacology
. 175:830-839
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7 .
Discovery of a Novel Inhibitor of the Hedgehog Signaling Pathway through Cell-based Compound Discovery and Target Prediction
저자
by
Bert Klebl
;
Hans R. Schöler
;
Herbert Waldmann
;
Matthias Baumann
;
Gisbert Schneider
, et al.
소스
Angewandte Chemie International Edition
. 56:13021-13025
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7 .
Systematic Kinase Inhibitor Profiling Identifies CDK9 as a Synthetic Lethal Target in NUT Midline Carcinoma
저자
by
Felix Dietlein
;
Roman K. Thomas
;
Martin Peifer
;
Daniel Rauh
;
Zoltán Varga
, et al.
소스
Cell Reports
Cell Reports, Vol 20, Iss 12, Pp 2833-2845 (2017)
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