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1 . Academic Journal
Indole Inhibitors of MMP-13 for Arthritic Disorders
저자
by
Steven J. Taylor
;
Asitha Abeywardane
;
Shuang Liang
;
Zhaoming Xiong
;
John R. Proudfoot
, et al.
소스
ACS Omega, Vol 6, Iss 29, Pp 18635-18650 (2021)
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7 .
Indole Inhibitors of MMP-13 for Arthritic Disorders
저자
by
John Xiang Li
;
Steven John Taylor
;
Mariana Margarit
;
Jun Li
;
Yu Yang
, et al.
소스
ACS Omega
ACS Omega, Vol 6, Iss 29, Pp 18635-18650 (2021)
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7 .
Discovery and optimization of oxadiazole-based FLAP inhibitors
저자
by
John D. Huber
;
J. Matthew Hutzler
;
Doris Riether
;
Tom Simpson
;
Alan Olague
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 27:4652-4659
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7 . Academic Journal
Fragment-Based Discoveryof Indole Inhibitors of MatrixMetalloproteinase-13.
저자
by
Steven J. Taylor
;
Asitha Abeywardane
;
Shuang Liang
;
Ingo Muegge
;
Anil K. Padyana
, et al.
소스
Journal of Medicinal Chemistry
. Dec2011, Vol. 54 Issue 23, p8174-8187. 14p.
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7 .
Synthesis, SAR, and Series Evolution of Novel Oxadiazole-Containing 5-Lipoxygenase Activating Protein Inhibitors: Discovery of 2-[4-(3-{(R)-1-[4-(2-Amino-pyrimidin-5-yl)-phenyl]-1-cyclopropyl-ethyl}-[1,2,4]oxadiazol-5-yl)-pyrazol-1-yl]-N,N-dimethyl-acetamide (BI 665915)
저자
by
Adam Flegg
;
Tina Morwick
;
Ho Yin Lo
;
Todd Bosanac
;
Weimin Liu
, et al.
소스
Journal of Medicinal Chemistry
. 58:1669-1690
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7 .
Discovery of Potent, Selective Chymase Inhibitors via Fragment Linking Strategies
저자
by
Xiang Li
;
Hidenori Takahashi
;
Steven S. Pullen
;
Stéphane De Lombaert
;
Asitha Abeywardane
, et al.
소스
Journal of Medicinal Chemistry
. 56:4465-4481
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7 .
Integrated strategies for identifying leads that target the NS3 helicase of the hepatitis C virus
저자
by
Anil Kumar Padyana
;
Xiang Li
;
Asitha Abeywardane
;
Pierre R. Bonneau
;
René Coulombe
, et al.
소스
Journal of medicinal chemistry
. 57(5)
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7 .
4+3 Cycloaddition reactions of halogen-substituted cyclohexenyl oxyallylic cations
저자
by
Michael Harmata
;
Asitha Abeywardane
;
László Kürti
;
Lixin Shao
.
소스
Tetrahedron Letters
. 40:1075-1078
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6 .
Correction to Fragment-Based Discovery of Indole Inhibitors of Matrix Metalloproteinase-13
저자
by
Zhaoming Xiong
;
Anil Kumar Padyana
;
John R. Proudfoot
;
Neil A. Farrow
;
Ingo Muegge
, et al.
소스
Journal of Medicinal Chemistry
. 58:6318-6318
Open Access (OpenAIRE)
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7 .
Fragment-based discovery of indole inhibitors of matrix metalloproteinase-13
저자
by
John Xiang Li
;
Xiang Li
;
Ingo Muegge
;
Steven John Taylor
;
Hani Zaher
, et al.
소스
Journal of medicinal chemistry
. 54(23)
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