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1 .
Synthesis and Anti-HCV Activity of Sugar-Modified Guanosine Analogues: Discovery of AL-611 as an HCV NS5B Polymerase Inhibitor for the Treatment of Chronic Hepatitis C
저자
by
Antitsa Dimitrova Stoycheva
;
Leonid Beigelman
;
Tongqian Chen
;
Kenneth Shaw
;
Vivek K. Rajwanshi
, et al.
소스
Journal of Medicinal Chemistry
. 63:10380-10395
Web of Science
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7 .
ALG-097111, a potent and selective SARS-CoV-2 3-chymotrypsin-like cysteine protease inhibitor exhibits in vivo efficacy in a Syrian Hamster model
저자
by
Leonid Beigelman
;
Jerome Deval
;
Lawrence M. Blatt
;
Dorothée Bardiot
;
Laura Vangeel
, et al.
소스
Biochemical and Biophysical Research Communications
Open Access (OpenAIRE)
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7 .
ALG-097111, a potent and selective SARS-CoV-2 3-chymotrypsin-like cysteine protease inhibitor exhibitsin vivoefficacy in a Syrian Hamster model
저자
by
Andreas Jekle
;
Julian A. Symons
;
Sushmita Mukherjee Chanda
;
Vladimir Serebryany
;
Leonid Beigelman
, et al.
소스
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7 .
Activation Pathway of a Nucleoside Analog Inhibiting Respiratory Syncytial Virus Polymerase
저자
by
Guangyi Wang
;
Yuen Tam
;
Antitsa Dimitrova Stoycheva
;
Jerome Deval
;
Sarah K. Stevens
, et al.
소스
ACS Chemical Biology
. 12:83-91
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7 .
Synthesis and Anti-HCV Activities of 4'-Fluoro-2'-Substituted Uridine Triphosphates and Nucleotide Prodrugs: Discovery of 4'-Fluoro-2'- C-methyluridine 5'-Phosphoramidate Prodrug (AL-335) for the Treatment of Hepatitis C Infection
저자
by
Yongfei Huang
;
Leonid Beigelman
;
Antitsa Dimitrova Stoycheva
;
Andreas Jekle
;
Zhinan Jin
, et al.
소스
Journal of medicinal chemistry
. 62(9)
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7 .
Regulation of gene transcription by thyroid hormone receptor β agonists in clinical development for the treatment of non-alcoholic steatohepatitis (NASH)
저자
by
Tse-I Lin
;
Lawrence M. Blatt
;
Andreas Jekle
;
Dinah Misner
;
Pierre Jean-Marie Bernard Raboisson
, et al.
소스
PLoS ONE
PLoS ONE, Vol 15, Iss 12, p e0240338 (2020)
Open Access (OpenAIRE)
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7 .
Abstract 4520: Preclinical characterization of ALG-031048, a novel STING agonist with potent anti-tumor activity in mice
저자
by
David Smith
;
April Kinkade
;
Sushmita Chanda
;
Antitsa Dimitrova Stoycheva
;
Dinah Misner
, et al.
소스
Cancer Research
. 80:4520-4520
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7 .
Abstract 1758: Discovery of novel potent and selective inhibitors of PRMT5 with anti-tumor activity in hepatocellular carcinoma and lung pre-clinical models
저자
by
Koen Vandyck
;
Antitsa Dimitrova Stoycheva
;
Francois Gonzalvez
;
Jyanwei Liu
;
Dinah Misner
, et al.
소스
Cancer Research
. 80:1758-1758
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7 .
HCV NS5B polymerase inhibitors 2: Synthesis and in vitro activity of (1,1-dioxo-2H-[1,2,4]benzothiadiazin-3-yl) azolo[1,5-a]pyridine and azolo[1,5-a]pyrimidine derivatives
저자
by
Antitsa Dimitrova Stoycheva
;
Leonid Beigelman
;
Karl Kossen
;
P. T. Ravi Rajagopalan
;
Donald Ruhrmund
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 19:4480-4483
Web of Science
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7 .
Preclinical Characteristics of the Hepatitis C Virus NS3/4A Protease Inhibitor ITMN-191 (R7227)
저자
by
Jin Hong
;
Christine Lemieux
;
Scott D. Seiwert
;
Shawn Misialek
;
Robert Rieger
, et al.
소스
Antimicrobial Agents and Chemotherapy
. 52:4432-4441
Full Text (ASM)
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