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1 . Academic Journal
Diacylglycerol acyltransferase-1 inhibition enhances intestinal fatty acid oxidation and reduces energy intake in rats[S]
저자
by
Gudrun Schober
;
Myrtha Arnold
;
Susan Birtles
;
Linda K. Buckett
;
Gustavo Pacheco-López
, et al.
소스
Journal of Lipid Research, Vol 54, Iss 5, Pp 1369-1384 (2013)
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7 . Academic Journal
Intestinal DGAT1 deficiency reduces postprandial triglyceride and retinyl ester excursions by inhibiting chylomicron secretion and delaying gastric emptying
저자
by
Gene P. Ables
;
Kryscilla Jian Zhang Yang
;
Silke Vogel
;
Antonio Hernandez-Ono
;
Shuiqing Yu
, et al.
소스
Journal of Lipid Research, Vol 53, Iss 11, Pp 2364-2379 (2012)
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7 . Academic Journal
DGAT1 deficiency decreases PPAR expression and does not lead to lipotoxicity in cardiac and skeletal muscle[S]
저자
by
Li Liu
;
Shuiqing Yu
;
Raffay S. Khan
;
Gene P. Ables
;
Kalyani G. Bharadwaj
, et al.
소스
Journal of Lipid Research, Vol 52, Iss 4, Pp 732-744 (2011)
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7 . Academic Journal
Discovery of a Potent, Selective, and Orally Efficacious Pyrimidinooxazinyl Bicyclooctaneacetic Acid Diacylglycerol Acyltransferase-1 Inhibitor.
저자
by
Alan M. Birch
;
Susan Birtles
;
Linda K. Buckett
;
Paul D. Kemmitt
;
Graham J. Smith
, et al.
소스
Journal of Medicinal Chemistry
. Mar2009, Vol. 52 Issue 6, p1558-1568. 11p.
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7 .
Translational Modeling to Guide Study Design and Dose Choice in Obesity Exemplified by AZD1979, a Melanin-concentrating Hormone Receptor 1 Antagonist
저자
by
Peter Gennemark
;
Daniel Lindén
;
Andrew V. Turnbull
;
Anders Johansson
;
Madeleine Antonsson
, et al.
소스
CPT: Pharmacometrics & Systems Pharmacology
. 6:458-468
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7 .
Effects of a novel potent melanin-concentrating hormone receptor 1 antagonist, AZD1979, on body weight homeostasis in mice and dogs
저자
by
Lillevi Kärrberg
;
Suzanne L. Iverson
;
Andrew V. Turnbull
;
Lambertus Benthem
;
Jenny Börjesson
, et al.
소스
British Journal of Pharmacology
. 173:2739-2751
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7 .
Novel role of a triglyceride-synthesizing enzyme
저자
by
Vinay Sachdev
;
Christina Leopold
;
Raimund Bauer
;
Jay V. Patankar
;
Jahangir Iqbal
, et al.
소스
ATHEROSCLEROSIS, 275, E10-E11. ELSEVIER IRELAND LTD
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7 .
Optimization of Brain Penetrant 11β-Hydroxysteroid Dehydrogenase Type I Inhibitors and in Vivo Testing in Diet-Induced Obese Mice
저자
by
Frederick W. Goldberg
;
Andrew V. Turnbull
;
Joanne deSchoolmeester
;
Martin Wild
;
Graeme R. Robb
, et al.
소스
Journal of Medicinal Chemistry
. 57:970-986
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7 .
11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Inhibitors Still Improve Metabolic Phenotype in Male 11β-HSD1 Knockout Mice Suggesting Off-Target Mechanisms
저자
by
Andrew V. Turnbull
;
Joanne deSchoolmeester
;
Pablo Morentin Gutierrez
;
Alice Yu
;
Elizabeth Cottrell
, et al.
소스
Endocrinology
Full Text (OUP)
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7 .
ACAT-selective and Nonselective DGAT1 Inhibition
저자
by
Tim J.D. Smith
;
Alan Martin Birch
;
Andrew V. Turnbull
;
Huw B. Jones
;
Linda K. Buckett
, et al.
소스
Toxicologic Pathology
. 41:941-950
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